BDBM50473228 AGN-190837::CHEMBL297752
SMILES CCC[C@H]1CCCC[C@@H]1NC1=NCCO1
InChI Key InChIKey=WDSZUSABLKNHCZ-QWRGUYRKSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50473228
Affinity DataKi: 3nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibitory constant determined using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 9.30nMAssay Description:Alpha-2B adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Alpha-2C adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Alpha-2A adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair