BDBM50498972 CHEMBL3735638
SMILES CC(C)n1c(C)nc2cnc(Nc3ccnc(n3)N3CCC(C)(C3)C(N)=O)cc12
InChI Key InChIKey=WPZKCOGUAMITHT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50498972
Affinity DataKi: 124nMAssay Description:Inhibition of human EGFR T790M/L858R double mutant using Fl-EEPLYWSFPAKKK-CONH2 as substrate preincubated for 30 mins followed by addition of substra...More data for this Ligand-Target Pair
Affinity DataKi: 681nMAssay Description:Inhibition of human wild type EGFR using Fl-EEPLYWSFPAKKK-CONH2 as substrate preincubated for 30 mins followed by addition of substrate measured afte...More data for this Ligand-Target Pair