BDBM74548 4-Amino-isothiazole-3,5-dicarboxylic acid 3-amide 5-[(tert-butylcarbamoyl-furan-2-yl-methyl)-(4-fluoro-benzyl)-amide]::4-amino-5-N-[2-(tert-butylamino)-1-(furan-2-yl)-2-oxoethyl]-5-N-[(4-fluorophenyl)methyl]-1,2-thiazole-3,5-dicarboxamide::4-amino-N'-[2-(tert-butylamino)-1-(2-furyl)-2-keto-ethyl]-N'-(4-fluorobenzyl)isothiazole-3,5-dicarboxamide::4-amino-N5-[2-(tert-butylamino)-1-(2-furanyl)-2-oxoethyl]-N5-[(4-fluorophenyl)methyl]isothiazole-3,5-dicarboxamide::4-azanyl-N5-[2-(tert-butylamino)-1-(furan-2-yl)-2-oxidanylidene-ethyl]-N5-[(4-fluorophenyl)methyl]-1,2-thiazole-3,5-dicarboxamide::MLS000072458::SMR000002677::cid_646665

SMILES CC(C)(C)NC(=O)C(N(Cc1ccc(F)cc1)C(=O)c1snc(C(N)=O)c1N)c1ccco1

InChI Key InChIKey=XUUFNGVDMWCRBB-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 74548   

TargetImportin subunit alpha-1(Homo sapiens (Human))
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM74548(4-Amino-isothiazole-3,5-dicarboxylic acid 3-amide ...)
Affinity DataEC50: >5.00E+5nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
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