BDBM7967 1-methyl-5-(beta-aminoethyl)-imidazole::2-(1-methyl-1H-imidazol-5-yl)ethan-1-amine::CHEMBL14722::L-histamine deriv. 1

SMILES Cn1cncc1CCN

InChI Key InChIKey=CPAGZVLINCPJEH-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 7967   

TargetHistamine H3 receptor(Rat)
Gliatech

Curated by ChEMBL
LigandPNGBDBM7967(1-methyl-5-(beta-aminoethyl)-imidazole | 2-(1-meth...)
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM7967(1-methyl-5-(beta-aminoethyl)-imidazole | 2-(1-meth...)
Affinity DataKi:  1.20E+5nMAssay Description:QC activity was evaluated fluorometrically using Gln-AMC as substrate, and pyroglutamyl peptidase as the auxiliary enzyme. After conversion of Gln-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed