BDBM8979 CHEMBL486901::N-[2-(1-benzylpiperidin-4-yl)ethyl]-2-(1,2,3,4-tetrahydroacridin-9-ylamino)acetamide::tacrine-E2020 analog 3
SMILES O=C(CNc1c2CCCCc2nc2ccccc12)NCCC1CCN(Cc2ccccc2)CC1
InChI Key InChIKey=AYESZVAJFBYQHK-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 8979
Affinity DataIC50: 6nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The appearance of product was monitored at 412 nm for 5 min us...More data for this Ligand-Target Pair
Affinity DataIC50: 76nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The appearance of product was monitored at 412 nm for 5 min us...More data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibition of rat serum butyrylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibition of rat serum BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of rat cortex homogenate acetylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of rat cortex AChEMore data for this Ligand-Target Pair