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Found 48 Enz. Inhib. hit(s) with Target = '2-oxoglutarate receptor 1'
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369952(CHEMBL609487)
Affinity DataKi:  10nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50409304(CHEMBL2113492)
Affinity DataKi:  12nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50409301(CHEMBL2092859)
Affinity DataKi:  12.9nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369155(CHEMBL609186)
Affinity DataKi:  17nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50409300(CHEMBL2113489)
Affinity DataKi:  18nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369942(CHEMBL607719)
Affinity DataKi:  19nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369943(CHEMBL608888)
Affinity DataKi:  20nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369937(CHEMBL608293)
Affinity DataKi:  20nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369938(CHEMBL1791423)
Affinity DataKi:  20nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369947(CHEMBL608296)
Affinity DataKi:  21nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369936(CHEMBL609773)
Affinity DataKi:  22nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369941(CHEMBL608893)
Affinity DataKi:  23nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369933(CHEMBL612154)
Affinity DataKi:  27nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369930(CHEMBL609776)
Affinity DataKi:  29nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369950(CHEMBL609769)
Affinity DataKi:  31nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50389796(CHEMBL1235128)
Affinity DataKi:  31nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  37nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  37nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369932(CHEMBL608595)
Affinity DataKi:  41nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM85777(B-NECA)
Affinity DataKi:  42nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369945(CHEMBL609775)
Affinity DataKi:  46nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50389799(CHEMBL2070508)
Affinity DataKi:  49nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50407975(CHEMBL519809)
Affinity DataKi:  51nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50409303(CHEMBL2092773)
Affinity DataKi:  55.6nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50409302(CHEMBL2113434)
Affinity DataKi:  58nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50367376(CHEMBL605866)
Affinity DataKi:  64nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369935(CHEMBL608587)
Affinity DataKi:  67nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369949(CHEMBL608591)
Affinity DataKi:  69.5nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50389798(CHEMBL2070507)
Affinity DataKi:  88nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50389797(CHEMBL261482)
Affinity DataKi:  96nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369944(CHEMBL609768)
Affinity DataKi:  123nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369928(CHEMBL608003)
Affinity DataKi:  140nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369946(CHEMBL609485)
Affinity DataKi:  163nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50106539((2S,3S,4R,5R)-5-(6-Amino-purin-9-yl)-3,4-dihydroxy...)
Affinity DataKi:  167nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369929(CHEMBL608895)
Affinity DataKi:  198nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369948(CHEMBL608596)
Affinity DataKi:  640nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369951(CHEMBL609179)
Affinity DataKi:  833nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369940(CHEMBL608000)
Affinity DataKi:  1.04E+3nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50369939(CHEMBL609774)
Affinity DataKi:  2.00E+3nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Rattus norvegicus)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50409305(CHEMBL2113436)
Affinity DataKi:  6.85E+3nMAssay Description:Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393123(CHEMBL2153446)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393148(CHEMBL2153586)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393117(CHEMBL2153440)
Affinity DataIC50:  7.00E+3nMAssay Description:Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393157(CHEMBL2153595)
Affinity DataIC50: >2.00E+4nMAssay Description:Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393161(CHEMBL2153439)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393129(CHEMBL2153461)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393143(CHEMBL2153581)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-oxoglutarate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393158(CHEMBL2153596)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed