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Compile Data Set for Download or QSAR

Marvin 2D Structure

Wt: 426.2
BDBM241108
Wt: 423.8
BDBM241126
Wt: 426.2
BDBM241138
Wt: 426.2
BDBM241139
Wt: 412.2
BDBM241140
Wt: 399.4
BDBM241141
Wt: 419.9
BDBM241146
Wt: 416.8
BDBM241155
Wt: 426.2
BDBM241158
Wt: 423.2
BDBM241098
Wt: 425.3
BDBM323242
Wt: 415.9
BDBM323243
Wt: 410.4
BDBM323245
Wt: 416.9
BDBM323249
Wt: 371.4
BDBM323252
Displayed 1 to 15 (of 80 total )  |  Next  |  Last  >>

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 25 hits in this display   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241108
PNG
(US9409895, 19 | US9630945, 19)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CCC(CC2)NC(=O)CCc2c[nH]nn2)c1
Show InChI InChI=1S/C18H21Cl2N5O3/c19-13-7-12(8-14(20)9-13)11-28-18(27)25-5-3-15(4-6-25)22-17(26)2-1-16-10-21-24-23-16/h7-10,15H,1-6,11H2,(H,22,26)(H,21,23,24)
PDB

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UniProtKB/SwissProt

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UniChem
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n/an/a 3n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241108
PNG
(US9409895, 19 | US9630945, 19)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CCC(CC2)NC(=O)CCc2c[nH]nn2)c1
Show InChI InChI=1S/C18H21Cl2N5O3/c19-13-7-12(8-14(20)9-13)11-28-18(27)25-5-3-15(4-6-25)22-17(26)2-1-16-10-21-24-23-16/h7-10,15H,1-6,11H2,(H,22,26)(H,21,23,24)
UniProtKB/SwissProt

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n/an/a 3n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241141
PNG
(US9409895, 51 | US9630945, 51)
Show SMILES Cc1cc(C)cc(COC(=O)N2CCC(CC2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C21H29N5O3/c1-15-10-16(2)12-17(11-15)14-29-21(28)26-8-6-18(7-9-26)23-20(27)5-3-4-19-13-22-25-24-19/h10-13,18H,3-9,14H2,1-2H3,(H,23,27)(H,22,24,25)
PDB

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Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241141
PNG
(US9409895, 51 | US9630945, 51)
Show SMILES Cc1cc(C)cc(COC(=O)N2CCC(CC2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C21H29N5O3/c1-15-10-16(2)12-17(11-15)14-29-21(28)26-8-6-18(7-9-26)23-20(27)5-3-4-19-13-22-25-24-19/h10-13,18H,3-9,14H2,1-2H3,(H,23,27)(H,22,24,25)
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n/an/a 6n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241146
PNG
(US9409895, 56 | US9630945, 56)
Show SMILES Cc1cc(Cl)cc(COC(=O)N2CCC(CC2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C20H26ClN5O3/c1-14-9-15(11-16(21)10-14)13-29-20(28)26-7-5-17(6-8-26)23-19(27)4-2-3-18-12-22-25-24-18/h9-12,17H,2-8,13H2,1H3,(H,23,27)(H,22,24,25)
PDB

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n/an/a 10n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241146
PNG
(US9409895, 56 | US9630945, 56)
Show SMILES Cc1cc(Cl)cc(COC(=O)N2CCC(CC2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C20H26ClN5O3/c1-14-9-15(11-16(21)10-14)13-29-20(28)26-7-5-17(6-8-26)23-19(27)4-2-3-18-12-22-25-24-18/h9-12,17H,2-8,13H2,1H3,(H,23,27)(H,22,24,25)
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n/an/a 10n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241140
PNG
(US9409895, 50 | US9630945, 50)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CC(C2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C17H19Cl2N5O3/c18-12-4-11(5-13(19)6-12)10-27-17(26)24-8-15(9-24)21-16(25)3-1-2-14-7-20-23-22-14/h4-7,15H,1-3,8-10H2,(H,21,25)(H,20,22,23)
PDB

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Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241140
PNG
(US9409895, 50 | US9630945, 50)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CC(C2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C17H19Cl2N5O3/c18-12-4-11(5-13(19)6-12)10-27-17(26)24-8-15(9-24)21-16(25)3-1-2-14-7-20-23-22-14/h4-7,15H,1-3,8-10H2,(H,21,25)(H,20,22,23)
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PC sid
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n/an/a 12n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM323245
PNG
(3-Cyano-5-methyl benzyl 4-(4-(1H-1,2,3-triazol-4-y...)
Show SMILES Cc1cc(COC(=O)N2CCC(CC2)NC(=O)CCCc2c[nH]nn2)cc(c1)C#N
Show InChI InChI=1S/C21H26N6O3/c1-15-9-16(12-22)11-17(10-15)14-30-21(29)27-7-5-18(6-8-27)24-20(28)4-2-3-19-13-23-26-25-19/h9-11,13,18H,2-8,14H2,1H3,(H,24,28)(H,23,25,26)
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n/an/a 13n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241155
PNG
(US9409895, 65 | US9630945, 65)
Show SMILES Clc1cc(COC(=O)N2CCC(CC2)NC(=O)CCc2c[nH]nn2)cc(c1)C#N
Show InChI InChI=1S/C19H21ClN6O3/c20-15-8-13(10-21)7-14(9-15)12-29-19(28)26-5-3-16(4-6-26)23-18(27)2-1-17-11-22-25-24-17/h7-9,11,16H,1-6,12H2,(H,23,27)(H,22,24,25)
PDB

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n/an/a 26n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241155
PNG
(US9409895, 65 | US9630945, 65)
Show SMILES Clc1cc(COC(=O)N2CCC(CC2)NC(=O)CCc2c[nH]nn2)cc(c1)C#N
Show InChI InChI=1S/C19H21ClN6O3/c20-15-8-13(10-21)7-14(9-15)12-29-19(28)26-5-3-16(4-6-26)23-18(27)2-1-17-11-22-25-24-17/h7-9,11,16H,1-6,12H2,(H,23,27)(H,22,24,25)
UniProtKB/SwissProt

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PC sid
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n/an/a 26n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM323249
PNG
(3-Chloro-5-cyanobenzyl 4-((4-(1H-1,2,3-triazol-4-y...)
Show SMILES Clc1cc(COC(=O)N2CCC(CC2)NCCCCc2c[nH]nn2)cc(c1)C#N
Show InChI InChI=1S/C20H25ClN6O2/c21-17-10-15(12-22)9-16(11-17)14-29-20(28)27-7-4-18(5-8-27)23-6-2-1-3-19-13-24-26-25-19/h9-11,13,18,23H,1-8,14H2,(H,24,25,26)
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n/an/a 29n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241138
PNG
(US9409895, 49 | US9630945, 49)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CCC(C2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C18H21Cl2N5O3/c19-13-6-12(7-14(20)8-13)11-28-18(27)25-5-4-16(10-25)22-17(26)3-1-2-15-9-21-24-23-15/h6-9,16H,1-5,10-11H2,(H,22,26)(H,21,23,24)
PDB

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n/an/a 48n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241138
PNG
(US9409895, 49 | US9630945, 49)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CCC(C2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C18H21Cl2N5O3/c19-13-6-12(7-14(20)8-13)11-28-18(27)25-5-4-16(10-25)22-17(26)3-1-2-15-9-21-24-23-15/h6-9,16H,1-5,10-11H2,(H,22,26)(H,21,23,24)
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n/an/a 48n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241126
PNG
(US9409895, 37 | US9630945, 37)
Show SMILES Fc1cc(Cl)cc(COC(=O)N2CCC(CC2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C19H23ClFN5O3/c20-14-8-13(9-15(21)10-14)12-29-19(28)26-6-4-16(5-7-26)23-18(27)3-1-2-17-11-22-25-24-17/h8-11,16H,1-7,12H2,(H,23,27)(H,22,24,25)
PDB

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n/an/a 55n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241126
PNG
(US9409895, 37 | US9630945, 37)
Show SMILES Fc1cc(Cl)cc(COC(=O)N2CCC(CC2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C19H23ClFN5O3/c20-14-8-13(9-15(21)10-14)12-29-19(28)26-6-4-16(5-7-26)23-18(27)3-1-2-17-11-22-25-24-17/h8-11,16H,1-7,12H2,(H,23,27)(H,22,24,25)
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n/an/a 55n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM323243
PNG
(3-Chloro-5-cyanobenzyl 4-(5-(1H-1,2,3-triazol-4-yl...)
Show SMILES Clc1cc(COC(=O)N2CCC(CCCCCc3c[nH]nn3)CC2)cc(c1)C#N
Show InChI InChI=1S/C21H26ClN5O2/c22-19-11-17(13-23)10-18(12-19)15-29-21(28)27-8-6-16(7-9-27)4-2-1-3-5-20-14-24-26-25-20/h10-12,14,16H,1-9,15H2,(H,24,25,26)
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n/an/a 69n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241098
PNG
(US9409895, 9 | US9630945, 9)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CCC(CC2)NC(=O)\C=C\c2c[nH]cn2)c1
Show InChI InChI=1S/C19H20Cl2N4O3/c20-14-7-13(8-15(21)9-14)11-28-19(27)25-5-3-16(4-6-25)24-18(26)2-1-17-10-22-12-23-17/h1-2,7-10,12,16H,3-6,11H2,(H,22,23)(H,24,26)/b2-1+
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Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241098
PNG
(US9409895, 9 | US9630945, 9)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CCC(CC2)NC(=O)\C=C\c2c[nH]cn2)c1
Show InChI InChI=1S/C19H20Cl2N4O3/c20-14-7-13(8-15(21)9-14)11-28-19(27)25-5-3-16(4-6-25)24-18(26)2-1-17-10-22-12-23-17/h1-2,7-10,12,16H,3-6,11H2,(H,22,23)(H,24,26)/b2-1+
PDB

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Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241139
PNG
(US9409895, 49b | US9630945, 49b)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CC[C@H](C2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C18H21Cl2N5O3/c19-13-6-12(7-14(20)8-13)11-28-18(27)25-5-4-16(10-25)22-17(26)3-1-2-15-9-21-24-23-15/h6-9,16H,1-5,10-11H2,(H,22,26)(H,21,23,24)/t16-/m1/s1
PDB

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Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241139
PNG
(US9409895, 49b | US9630945, 49b)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CC[C@H](C2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C18H21Cl2N5O3/c19-13-6-12(7-14(20)8-13)11-28-18(27)25-5-4-16(10-25)22-17(26)3-1-2-15-9-21-24-23-15/h6-9,16H,1-5,10-11H2,(H,22,26)(H,21,23,24)/t16-/m1/s1
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US Patent
n/an/a 263n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM323242
PNG
(3,5-Dichlorobenzyl 4-(5-(1H-1,2,3-triazol-4-yl)pen...)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CCC(CCCCCc3c[nH]nn3)CC2)c1
Show InChI InChI=1S/C20H26Cl2N4O2/c21-17-10-16(11-18(22)12-17)14-28-20(27)26-8-6-15(7-9-26)4-2-1-3-5-19-13-23-25-24-19/h10-13,15H,1-9,14H2,(H,23,24,25)
UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a 318n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2


(Homo sapiens (Human))
BDBM241158
PNG
(US9409895, 49a | US9630945, 49a)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CC[C@@H](C2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C18H21Cl2N5O3/c19-13-6-12(7-14(20)8-13)11-28-18(27)25-5-4-16(10-25)22-17(26)3-1-2-15-9-21-24-23-15/h6-9,16H,1-5,10-11H2,(H,22,26)(H,21,23,24)/t16-/m0/s1
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a>1.00E+3n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9409895 (2016)


BindingDB Entry DOI: 10.7270/Q2GT5M2G
More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM241158
PNG
(US9409895, 49a | US9630945, 49a)
Show SMILES Clc1cc(Cl)cc(COC(=O)N2CC[C@@H](C2)NC(=O)CCCc2c[nH]nn2)c1
Show InChI InChI=1S/C18H21Cl2N5O3/c19-13-6-12(7-14(20)8-13)11-28-18(27)25-5-4-16(10-25)22-17(26)3-1-2-15-9-21-24-23-15/h6-9,16H,1-5,10-11H2,(H,22,26)(H,21,23,24)/t16-/m0/s1
UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a>1.00E+3n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair
Ataxin-2


(Homo sapiens (Human))
BDBM323252
PNG
(US9630945, 78)
Show SMILES O=C(CCCc1c[nH]nn1)NC1CCN(CC1)C(=O)OCc1ccccc1
Show InChI InChI=1S/C19H25N5O3/c25-18(8-4-7-17-13-20-23-22-17)21-16-9-11-24(12-10-16)19(26)27-14-15-5-2-1-3-6-15/h1-3,5-6,13,16H,4,7-12,14H2,(H,21,25)(H,20,22,23)
UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a 1.39E+3n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...


US Patent US9630945 (2017)

More data for this
Ligand-Target Pair