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Found 13 Enz. Inhib. hit(s) with Target = 'Cytosolic beta-glucosidase'
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50383315(CHEMBL2029773)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human cytosolic beta-glucosidase using 4-methylumbelliferyl beta-D-glucopyranoside as substrate after 15 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50163441((2R,3S,4S,5R)-2-Hydroxymethyl-piperidine-3,4,5-tri...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibitory concentration against beta-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50163441((2R,3S,4S,5R)-2-Hydroxymethyl-piperidine-3,4,5-tri...)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibitory concentration against human beta-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibitory concentration against beta-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50:  2.40E+5nMAssay Description:Inhibitory concentration against human beta-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50234564(CHEMBL259905)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of beta-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50163447((2S,3S,4S,5R)-2-Hydroxymethyl-piperidine-3,4,5-tri...)
Affinity DataIC50:  9.80E+5nMAssay Description:Inhibitory concentration against beta-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50153476(4-((3R,8S)-4-Hydroxy-3-methoxy-6-oxa-bicyclo[3.2.1...)
Affinity DataIC50: <1.00E+6nMAssay Description:Inhibition of Beta-glucosidase of rat intestine; no inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50118923((1S,2S,3R)-4-Methyl-6-octylamino-cyclohexane-1,2,3...)
Affinity DataIC50: <1.00E+6nMAssay Description:Inhibition of Beta-glucosidase of rat intestine; no inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50153475(4-Hydroxymethyl-6-octylamino-cyclohexane-1,2,3-tri...)
Affinity DataIC50: <1.00E+6nMAssay Description:Inhibition of Beta-glucosidase of rat intestine; no inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50153474(4-Methylene-6-octylamino-cyclohexane-1,2,3-triol |...)
Affinity DataIC50: <1.00E+6nMAssay Description:Inhibition of Beta-glucosidase of rat intestine; no inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50153478(CHEMBL185536 | N-(2,3,4-Trihydroxy-5-hydroxymethyl...)
Affinity DataIC50:  1.40E+10nMAssay Description:Inhibition of Beta-glucosidase of rat intestineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50367332(CHEMBL1628264)
Affinity DataIC50:  1.30E+11nMAssay Description:Inhibition of Beta-glucosidase of rat intestineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed