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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
Monomer List in csv
Het List in SDF
Compound
FDA Drugs
Important Compounds
Chemical Structure
Name
SMILES
Number of Data
/
Targets
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3D Structure Series
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Author
Journal/Citation
Institution
PubMed
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Special Data Sets
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Prot-Lig Validation Sets
Other Databases
PDB
85%
100%
Seq ID
UniProtKB/Swiss-Prot
UniProtKB/TrEMBL
PubMed
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All Compounds & Data
Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Deposition
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cAMP-Dependent Protein Kinase (PKA)
List of PDBs
1CDK
1CMK
1CTP
1FMO
1J3H
1JBP
1JLU
1L3R
1Q24
1Q61
1Q62
1Q8T
1Q8U
1Q8W
1RDQ
1RE8
1REJ
1REK
1SMH
1STC
1SVE
1SVG
1SVH
1SYK
1SZM
1VEB
1XH4
1XH5
1XH6
1XH7
1XH8
1XH9
1XHA
1YDR
1YDS
1YDT
2C1A
2C1B
2CPK
2ERZ
2F7E
2F7X
2F7Z
2GFC
2GNF
2GNG
2GNH
2GNI
2GNJ
2GNL
2GU8
2JDS
2JDT
2JDV
2OH0
2OJF
2QCS
2QUR
2QVS
2UVX
2UVY
2UVZ
2UW0
2UW3
2UW4
2UW5
2UW6
2UW7
2UW8
2UZT
2UZU
2UZV
2UZW
2VNW
2VNY
2VO0
2VO3
2VO6
2VO7
3AG9
3AGL
3AGM
3AMA
3AMB
3BWJ
3DND
3DNE
3E8C
3E8E
3FHI
3FJQ
3IDB
3IDC
3J4Q
3J4R
3KKV
3L9L
3L9M
3L9N
3MVJ
3NX8
3O7L
3OOG
3OVV
3OW3
3OWP
3OXT
3P0M
3POO
3PVB
3QAL
3QAM
3TNP
3TNQ
3VQH
3X2U
3X2V
3X2W
3ZO1
3ZO2
3ZO3
3ZO4
4AE6
4AE9
4AXA
4C33
4C34
4C35
4C36
4C37
4C38
4DFX
4DFY
4DFZ
4DG0
4DG2
4DG3
4DH1
4DH3
4DH5
4DH7
4DH8
4DIN
4HPT
4HPU
4IAC
4IAD
4IAF
4IAI
4IAK
4IAY
4IAZ
4IB0
4IB1
4IB3
4IE9
4IJ9
4NTS
4NTT
4O21
4O22
4UJ1
4UJ2
4UJ9
4UJA
4UJB
4WB5
4WB6
4WB7
4WB8
4WBB
4WIH
4X6Q
4X6R
4XW4
4XW5
4XW6
4YXR
4YXS
4Z83
4Z84
5BX6
5BX7
5IZF
5IZJ
5J5X
5JR7
5LCP
5LCQ
5LCR
5LCT
5LCU
5M0B
5M0C
5M0L
5M0U
5M6V
5M6Y
5M71
5M75
5MHI
5N1D
5N1E
5N1F
5N1G
5N1H
5N1K
5N1L
5N1M
5N1N
5N1O
5N23
5N32
5N33
5N36
5N37
5N39
5N3A
5N3B
5N3C
5N3D
5N3E
5N3F
5N3G
5N3H
5N3I
5N3J
5N3K
5N3L
5N3M
5N3N
5N3O
5N3P
5N3Q
5N3R
5N3S
5N3T
5N7P
5N7U
5NTJ
5NW8
5O0E
5O5M
5OK3
5OL3
5OT3
5OTG
5OUA
5OUC
5OUS
5UZK
5VHB
5VI9
5VIB
5X3F
6BYR
6BYS
6C0U
6E21
6E99
6E9L
6EGW
6EH0
6EH2
6EH3
6EM2
6EM6
6EM7
6EMA
6EMB
6EMD
6ERS
6ERT
6ERU
6ERV
6ERW
6ESA
6F14
6FRX
6I2A
6I2B
6I2C
6I2D
6I2H
6MM5
6MM6
6MM7
6MM8
6NO7
6QJ7
6SNN
6SNX
6SOX
6SPM
6SPS
6SPU
6SPY
6SQ1
6WJF
6WJG