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Found 48 with Last Name = 'addlagatta' and Initial = 'a'
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50078539(CHEMBL3414950)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of Human MetAP1b using Met-pNA as substrateMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50337147((RS)-1-amino-3-cyclohexylpropylphosphonic acid | C...)
Affinity DataKi:  9.90E+3nMAssay Description:Inhibition of Human MetAP1b using Met-pNA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50078540(CHEMBL1673077)
Affinity DataKi:  5.48E+4nMAssay Description:Inhibition of Human MetAP1b using Met-pNA as substrateMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316031(CHEMBL1090366 | amino(phenyl)methylphosphonic acid)
Affinity DataKi:  1.12E+5nMAssay Description:Inhibition of Human MetAP1b using Met-pNA as substrateMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50078541(CHEMBL3414949)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of Human MetAP1b using Met-pNA as substrateMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50337150((RS)-1-amino-2-cyclohexylethylphosphonic acid | CH...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of Human MetAP1b using Met-pNA as substrateMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM17847(CHEMBL327579 | pyridine-2-carboxylic acid inhibito...)
Affinity DataIC50:  1.50E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499710(CHEMBL516021)
Affinity DataIC50:  1.79E+3nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50277158(3123L | CHEBI:17939 | CL-13900 | GNF-Pf-2016 | P-6...)
Affinity DataIC50:  2.45E+3nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM17849(3-(2,2-dimethylpropanamido)-N-(1,3-thiazol-2-yl)py...)
Affinity DataIC50:  2.90E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM17850(3-(3-phenylpropanamido)-N-(1,3-thiazol-2-yl)pyridi...)
Affinity DataIC50:  3.50E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM17851(3-[(E)-(2-methylpropylidene)amino]-N-(1,3-thiazol-...)
Affinity DataIC50:  6.40E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50062530(CHEMBL3397584)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499702(CHEMBL3740370)
Affinity DataIC50:  8.04E+3nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50062531(CHEMBL3397585)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499709(CHEMBL3741560)
Affinity DataIC50:  8.53E+3nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499705(CHEMBL3741724)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499712(CHEMBL3741833)
Affinity DataIC50:  3.27E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499707(CHEMBL3741904)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499708(CHEMBL3739649)
Affinity DataIC50:  3.64E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499706(CHEMBL3740199)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499704(CHEMBL3740158)
Affinity DataIC50:  6.88E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499713(CHEMBL3741344)
Affinity DataIC50:  8.10E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499701(CHEMBL3741701)
Affinity DataIC50:  9.25E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499703(CHEMBL3740862)
Affinity DataIC50:  9.29E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPuromycin-sensitive aminopeptidase(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499711(CHEMBL3741419)
Affinity DataIC50:  9.82E+4nMAssay Description:Inhibition of recombinant human puromycin sensitive aminopeptidase using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499709(CHEMBL3741560)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50277158(3123L | CHEBI:17939 | CL-13900 | GNF-Pf-2016 | P-6...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499706(CHEMBL3740199)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499705(CHEMBL3741724)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499704(CHEMBL3740158)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499708(CHEMBL3739649)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499707(CHEMBL3741904)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499703(CHEMBL3740862)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499702(CHEMBL3740370)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499701(CHEMBL3741701)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499710(CHEMBL516021)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499713(CHEMBL3741344)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499712(CHEMBL3741833)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50499711(CHEMBL3741419)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine aminopeptidase-N using Leu-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Johns Hopkins University

LigandPNGBDBM17847(CHEMBL327579 | pyridine-2-carboxylic acid inhibito...)
Affinity DataIC50: >3.00E+5nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Johns Hopkins University

LigandPNGBDBM17850(3-(3-phenylpropanamido)-N-(1,3-thiazol-2-yl)pyridi...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM17852(3-octanamido-N-(1,3-thiazol-2-yl)pyridine-2-carbox...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Johns Hopkins University

LigandPNGBDBM17852(3-octanamido-N-(1,3-thiazol-2-yl)pyridine-2-carbox...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Johns Hopkins University

LigandPNGBDBM17849(3-(2,2-dimethylpropanamido)-N-(1,3-thiazol-2-yl)py...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Johns Hopkins University

LigandPNGBDBM17851(3-[(E)-(2-methylpropylidene)amino]-N-(1,3-thiazol-...)
Affinity DataIC50: >1.00E+6nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Rattus norvegicus)
Tm Bhagalpur University

Curated by ChEMBL
LigandPNGBDBM50507632(CHEMBL4448381)
Affinity DataIC50:  3.13E+6nMAssay Description:Anti-biofilm activity against Enterococcus faecalis after 24 hrs by XTT assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed