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Found 63 with Last Name = 'agabiti' and Initial = 'ss'
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  4.56E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516697(CHEMBL4302450)
Affinity DataIC50:  7.87E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516697(CHEMBL4302450)
Affinity DataIC50:  7.87E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  9.64E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.21E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.61E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) at pH ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.61E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.61E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.65E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.99E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  2.30E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516698(CHEMBL4116247)
Affinity DataIC50:  1.03E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516699(CHEBI:16057 | DIMETHYLALLYL DIPHOSPHATE | Dimethyl...)
Affinity DataIC50:  2.70E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50: >3.33E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 H381R mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM25257(({hydroxy[(3-methylbut-3-en-1-yl)oxy]phosphoryl}ox...)
Affinity DataIC50:  5.13E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  1.04E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  1.07E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50278316(CHEMBL450079 | sodium pyrophosphate(V))
Affinity DataIC50:  1.14E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  2.56E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.19E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.22E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  3.24E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.39E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 M424A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  3.43E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  3.72E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.83E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.85E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.93E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  4.62E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  5.35E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 M424A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516698(CHEMBL4116247)
Affinity DataKd:  1.11E+5nMAssay Description:Binding affinity to C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) by isothermal calo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236895(CHEMBL4088948)
Affinity DataEC50:  5.40nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated cell proliferation by measuring increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataEC50:  3.40E+3nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated IFNgamma production measured after 48 hrs ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516699(CHEBI:16057 | DIMETHYLALLYL DIPHOSPHATE | Dimethyl...)
Affinity DataEC50:  1.50E+3nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated IFNgamma production measured after 48 hrs ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236889(CHEMBL4061531)
Affinity DataEC50:  41nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated cell proliferation by measuring increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM25257(({hydroxy[(3-methylbut-3-en-1-yl)oxy]phosphoryl}ox...)
Affinity DataEC50:  3.60E+4nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated cell proliferation by measuring increase i...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236895(CHEMBL4088948)
Affinity DataEC50:  15nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated IFNgamma production measured after 48 hrs ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM25257(({hydroxy[(3-methylbut-3-en-1-yl)oxy]phosphoryl}ox...)
Affinity DataEC50:  7.10E+4nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated IFNgamma production measured after 48 hrs ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataKd:  4.27E+3nMAssay Description:Binding affinity to C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) by isothermal calorimetric ti...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516698(CHEMBL4116247)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated IFNgamma production measured after 48 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516697(CHEMBL4302450)
Affinity DataEC50:  2nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated IFNgamma production measured after 48 hrs ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataEC50:  4.20nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated IFNgamma production measured after 48 hrs ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataEC50:  4.00E+3nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated cell proliferation by measuring increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516698(CHEMBL4116247)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated cell proliferation by measuring increase i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516697(CHEMBL4302450)
Affinity DataEC50:  86nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated cell proliferation by measuring increase i...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataEC50:  0.510nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated cell proliferation by measuring increase i...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236889(CHEMBL4061531)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated IFNgamma production measured after 48 hrs ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataKd:  1.54E+3nMAssay Description:Binding affinity to C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) by isothermal calo...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataEC50:  0.510nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataEC50:  4.00E+3nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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