Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human ChemR23 expressed in CAL-1 cells assessed as reduction in chemerin-induced calcium signalingMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10nMAssay Description:Inhibition of human ChemR23 expressed in CAL-1 cells assessed as reduction in chemerin-induced calcium signalingMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human ChemR23 expressed in CAL-1 cells assessed as reduction in chemerin-induced calcium signalingMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of human ChemR23 expressed in CAL-1 cells assessed as reduction in chemerin-induced calcium signalingMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human ChemR23 expressed in CAL-1 cells assessed as reduction in chemerin-induced calcium signalingMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human ChemR23 expressed in CAL-1 cells assessed as reduction in chemerin-induced calcium signalingMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Zeria Pharmaceutical
Curated by ChEMBL
Zeria Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase from Dawley rat prostateMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human ChemR23 expressed in CAL-1 assessed as increase in calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at human ChemR23 expressed in CAL-1 assessed as increase in calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Agonist activity at human ChemR23 expressed in CAL-1 assessed as increase in calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Inhibition of human ChemR23 expressed in CAL-1 cells assessed as receptor internalizationMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Agonist activity at human ChemR23 expressed in CAL-1 assessed as increase in calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Agonist activity at human ChemR23 expressed in CAL-1 assessed as increase in calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Agonist activity at human ChemR23 expressed in CAL-1 assessed as increase in calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Agonist activity at human ChemR23 expressed in CAL-1 assessed as increase in calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at human ChemR23 expressed in CAL-1 assessed as increase in calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Inhibition of human ChemR23 expressed in CAL-1 cells assessed as receptor internalizationMore data for this Ligand-Target Pair
Affinity DataEC50: 440nMAssay Description:Agonist activity at human ChemR23 expressed in CAL-1 assessed as increase in calcium mobilizationMore data for this Ligand-Target Pair