Affinity DataIC50: <0.400nMAssay Description:Inhibition of human MAGLMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Inhibition of human MAGL transfected in human HEK293T cells assessed as reduction in ABPP binding by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 117nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human Jurkat cell membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 151nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 196nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 242nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 282nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 424nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 815nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.85E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.05E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.06E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.19E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.19E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 3.77E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair