Compile Data Set for Download or QSAR
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Found 260 with Last Name = 'akssira' and Initial = 'm'
TargetDihydrofolate reductase(Pneumocystis carinii)
Universit£

Curated by ChEMBL
LigandPNGBDBM50135141(6-[(2,5-Dichloro-phenylamino)-methyl]-pyrido[2,3-d...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of recombinant Pneumocystis carinii DHFR expressed in Escherichia coli Rosetta Gami B (DE3) by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50135141(6-[(2,5-Dichloro-phenylamino)-methyl]-pyrido[2,3-d...)
Affinity DataKi:  24nMAssay Description:Inhibition of recombinant human DHFR expressed in Escherichia coli Rosetta Gami B (DE3) by spectrophotometric assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50243145(CHEMBL3109141)
Affinity DataIC50:  1nMAssay Description:Inhibition of mTOR (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50094703(5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataIC50:  2nMAssay Description:Inhibition of adenosine kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50495494(CHEMBL3109116)
Affinity DataIC50:  3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50243143(CHEMBL3109142)
Affinity DataIC50:  5nMAssay Description:Inhibition of mTOR (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50099963(CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...)
Affinity DataIC50:  7nMAssay Description:Inhibition of EGFR intracellular domain (unknown origin) purified from a baculovirus expression system using Biotin-(amino hexonoic acid)-EEEEYFELVAK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50495487(CHEMBL3109134)
Affinity DataIC50:  7nMAssay Description:Inhibition of PI3Kalpha (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50495501(CHEMBL3109133)
Affinity DataIC50:  8nMAssay Description:Inhibition of PI3Kdelta (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50495499(CHEMBL3109140)
Affinity DataIC50:  13nMAssay Description:Inhibition of mTOR (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50243143(CHEMBL3109142)
Affinity DataIC50:  14nMAssay Description:Inhibition of PI3Kdelta (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50099963(CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...)
Affinity DataIC50:  16nMAssay Description:Inhibition of ErbB-2 intracellular domain (unknown origin) purified from a baculovirus expression system using Biotin-(amino hexonoic acid)-EEEEYFELV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional dihydrofolate reductase-thymidylate synthase(Toxoplasma gondii)
Universit£

Curated by ChEMBL
LigandPNGBDBM18224(6-[(2,5-dimethoxyphenyl)methyl]-5-methylpyrido[2,3...)
Affinity DataIC50:  17nMAssay Description:Inhibition of Toxoplasma gondii DHFR by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50495491(CHEMBL3109139)
Affinity DataIC50:  18nMAssay Description:Inhibition of PI3Kdelta (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50495494(CHEMBL3109116)
Affinity DataIC50:  19nMAssay Description:Inhibition of PI3Kalpha (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Pneumocystis carinii)
Universit£

Curated by ChEMBL
LigandPNGBDBM18224(6-[(2,5-dimethoxyphenyl)methyl]-5-methylpyrido[2,3...)
Affinity DataIC50:  19nMAssay Description:Inhibition of Pneumocystis carinii DHFR by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50073942(CHEMBL3409483)
Affinity DataIC50:  21nMAssay Description:Inhibition of ErbB-2 intracellular domain (unknown origin) purified from a baculovirus expression system using Biotin-(amino hexonoic acid)-EEEEYFELV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50073942(CHEMBL3409483)
Affinity DataIC50:  23nMAssay Description:Inhibition of EGFR intracellular domain (unknown origin) purified from a baculovirus expression system using Biotin-(amino hexonoic acid)-EEEEYFELVAK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50161356(CHEMBL3786536)
Affinity DataIC50:  23nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50495514(CHEMBL3109126)
Affinity DataIC50:  24nMAssay Description:Inhibition of PI3Kdelta (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50161347(CHEMBL3786624)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50073941(CHEMBL3409484)
Affinity DataIC50:  25nMAssay Description:Inhibition of EGFR intracellular domain (unknown origin) purified from a baculovirus expression system using Biotin-(amino hexonoic acid)-EEEEYFELVAK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399310(CHEMBL2180854)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50073941(CHEMBL3409484)
Affinity DataIC50:  26nMAssay Description:Inhibition of ErbB-2 intracellular domain (unknown origin) purified from a baculovirus expression system using Biotin-(amino hexonoic acid)-EEEEYFELV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243143(CHEMBL3109142)
Affinity DataIC50:  26nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50495501(CHEMBL3109133)
Affinity DataIC50:  27nMAssay Description:Inhibition of PI3Kalpha (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50495487(CHEMBL3109134)
Affinity DataIC50:  29nMAssay Description:Inhibition of PI3Kdelta (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50073943(CHEMBL3409482)
Affinity DataIC50:  30nMAssay Description:Inhibition of ErbB-2 intracellular domain (unknown origin) purified from a baculovirus expression system using Biotin-(amino hexonoic acid)-EEEEYFELV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50495494(CHEMBL3109116)
Affinity DataIC50:  31nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50495498(CHEMBL3109146)
Affinity DataIC50:  35nMAssay Description:Inhibition of mTOR (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50161348(CHEMBL3785408)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50495485(CHEMBL3109143)
Affinity DataIC50:  36nMAssay Description:Inhibition of mTOR (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50073943(CHEMBL3409482)
Affinity DataIC50:  36nMAssay Description:Inhibition of EGFR intracellular domain (unknown origin) purified from a baculovirus expression system using Biotin-(amino hexonoic acid)-EEEEYFELVAK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50495494(CHEMBL3109116)
Affinity DataIC50:  37nMAssay Description:Inhibition of mTOR (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399303(CHEMBL2180844)
Affinity DataIC50:  37nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399312(CHEMBL2180852)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50161338(CHEMBL3787480)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243145(CHEMBL3109141)
Affinity DataIC50:  40nMAssay Description:Inhibition of PI3Kalpha (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50161339(CHEMBL3787512)
Affinity DataIC50:  41nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50161398(CHEMBL3787292)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50161345(CHEMBL3785575)
Affinity DataIC50:  44nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50495486(CHEMBL3109144)
Affinity DataIC50:  45nMAssay Description:Inhibition of PI3Kalpha (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50495498(CHEMBL3109146)
Affinity DataIC50:  45nMAssay Description:Inhibition of PI3Kalpha (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50495486(CHEMBL3109144)
Affinity DataIC50:  54nMAssay Description:Inhibition of mTOR (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50243143(CHEMBL3109142)
Affinity DataIC50:  58nMAssay Description:Inhibition of PI3Kalpha (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50495487(CHEMBL3109134)
Affinity DataIC50:  59nMAssay Description:Inhibition of mTOR (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50495497(CHEMBL3109115)
Affinity DataIC50:  59nMAssay Description:Inhibition of PI3Kalpha (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50495514(CHEMBL3109126)
Affinity DataIC50:  61nMAssay Description:Inhibition of PI3Kalpha (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50243145(CHEMBL3109141)
Affinity DataIC50:  62nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50161344(CHEMBL3786276)
Affinity DataIC50:  67nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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