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Found 47 with Last Name = 'almeida' and Initial = 's'
TargetBeta-galactosidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50469238(CHEMBL4288931)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of beta-galactosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-galactopyranoside as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556691(CHEMBL4760140)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-galactosidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235812(CHEMBL4085739)
Affinity DataIC50:  10nMAssay Description:Inhibition of beta-galactosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-galactopyranoside as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-galactosidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50469239(CHEMBL4284436)
Affinity DataIC50:  10nMAssay Description:Inhibition of beta-galactosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-galactopyranoside as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50376383(CHEMBL259972)
Affinity DataIC50:  13nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50182801((3R,4R,5R)-5-(Hydroxymethyl)piperidine-3,4-diol, 8...)
Affinity DataIC50:  20nMAssay Description:Inhibition of beta-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-glucopyranoside as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50469238(CHEMBL4288931)
Affinity DataIC50:  40nMAssay Description:Inhibition of beta-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-glucopyranoside as subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556695(CHEMBL4746714)
Affinity DataIC50:  50nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556696(CHEMBL4759732)
Affinity DataIC50:  75nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556690(CHEMBL4799478)
Affinity DataIC50:  80nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556697(CHEMBL4789403)
Affinity DataIC50:  90nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556685(CHEMBL4740788)
Affinity DataIC50:  120nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556688(CHEMBL4744394)
Affinity DataIC50:  150nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50469275(CHEMBL4290673)
Affinity DataIC50:  180nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-galactosidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50469237(CHEMBL4281031)
Affinity DataIC50:  250nMAssay Description:Inhibition of beta-galactosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-galactopyranoside as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50469275(CHEMBL4290673)
Affinity DataIC50:  250nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human COX-2 expressed in Baculovirus infected Sf21 cells using arachidonic acid as substrate preincu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  260nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human COX-2 expressed in Baculovirus infected Sf21 cells using arachidonic acid as substrate preincu...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556696(CHEMBL4759732)
Affinity DataIC50:  300nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556694(CHEMBL4758894)
Affinity DataIC50:  500nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556693(CHEMBL4794474)
Affinity DataIC50:  800nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556692(CHEMBL4789452)
Affinity DataIC50:  950nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50469276(CHEMBL4282782)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human COX-2 expressed in Baculovirus infected Sf21 cells using arachidonic acid as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50469276(CHEMBL4282782)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  3.09E+3nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556692(CHEMBL4789452)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556685(CHEMBL4740788)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556687(CHEMBL4788569)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556686(CHEMBL4749219)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235812(CHEMBL4085739)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of beta-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-glucopyranoside as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50469239(CHEMBL4284436)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of beta-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-glucopyranoside as subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-galactosidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50182801((3R,4R,5R)-5-(Hydroxymethyl)piperidine-3,4-diol, 8...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of beta-galactosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-galactopyranoside as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50469237(CHEMBL4281031)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of beta-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-glucopyranoside as subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556693(CHEMBL4794474)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556697(CHEMBL4789403)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556694(CHEMBL4758894)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556687(CHEMBL4788569)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556688(CHEMBL4744394)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556689(CHEMBL4791495)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556690(CHEMBL4799478)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50376383(CHEMBL259972)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556686(CHEMBL4749219)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556691(CHEMBL4760140)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556695(CHEMBL4746714)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human COX-2 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50556689(CHEMBL4791495)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX-1 assessed as peroxidase activity using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50469238(CHEMBL4288931)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl alpha-D-glucopyranoside as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50235812(CHEMBL4085739)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl alpha-D-glucopyranoside as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50469237(CHEMBL4281031)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl alpha-D-glucopyranoside as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed