Compile Data Set for Download or QSAR
maximum 50k data
Found 100 with Last Name = 'amendt' and Initial = 'c'
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313441(3-(dimethylamino)-N-(((2R,4aS,5R,10bS)-9-isopropyl...)
Affinity DataIC50:  2nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313446(CHEMBL1096003 | N-(((2R,4aS,5R,10bS)-9-chloro-7-fl...)
Affinity DataIC50:  2nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313442(1-((2R,4aS,5R,10bS)-9-bromo-7-fluoro-5-phenyl-3,4,...)
Affinity DataIC50:  3nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313437(1-((2R,4aS,5R,10bS)-9-tert-butyl-5-phenyl-3,4,4a,5...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313435(4-((2R,4aS,5R,10bS)-2-((methylamino)methyl)-9-(tri...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313430(2-(methylamino)-N-(((2R,4aS,5R,10bS)-5-phenyl-9-(t...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313444(CHEMBL1085692 | N-(((2R,4aS,5R,10bS)-9-bromo-7-flu...)
Affinity DataIC50:  5nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313439(1-((2R,4aS,5R,10bS)-9-tert-butyl-5-(thiophen-2-yl)...)
Affinity DataIC50:  5nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313434((2R,4aS,5R,10bS)-2-((1H-1,2,4-triazol-1-yl)methyl)...)
Affinity DataIC50:  6nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313443(CHEMBL1082249 | N-(2-(((2R,4aS,5R,10bS)-9-bromo-7-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313445(2-(((2R,4aS,5R,10bS)-9-chloro-7-fluoro-5-phenyl-3,...)
Affinity DataIC50:  7nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313431(3-amino-N-methyl-N-(((2R,4aS,5R,10bS)-5-phenyl-9-(...)
Affinity DataIC50:  7nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313428(1-(2-(dimethylamino)ethyl)-3-(((2R,4aS,5R,10bS)-5-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313427(1-(3-hydroxypropyl)-3-(((2R,4aS,5R,10bS)-5-phenyl-...)
Affinity DataIC50:  11nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313440(1-((2R,4aS,5R,10bS)-9-cyclopropyl-5-phenyl-3,4,4a,...)
Affinity DataIC50:  11nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313429(2-(dimethylamino)ethyl((2R,4aS,5R,10bS)-5-phenyl-9...)
Affinity DataIC50:  14nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313409(4-((4aS,5R,10bS)-9-tert-butyl-3,4,4a,5,6,10b-hexah...)
Affinity DataIC50:  17nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313432(CHEMBL1093087 | N1-phenyl-N1-(((2R,4aS,5R,10bS)-5-...)
Affinity DataIC50:  19nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313438(2-((((2R,4aS,5R,10bS)-9-tert-butyl-5-phenyl-3,4,4a...)
Affinity DataIC50:  19nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313426(((2R,4aS,5R,10bS)-5-phenyl-9-(trifluoromethyl)-3,4...)
Affinity DataIC50:  20nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313418((4aS,5R,10bS)-9-tert-butyl-5-(thiophen-2-yl)-3,4,4...)
Affinity DataIC50:  25nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313407(4-((4aS,5R,10bS)-9-tert-butyl-3,4,4a,5,6,10b-hexah...)
Affinity DataIC50:  34nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313406(3-((4aS,5R,10bS)-9-tert-butyl-3,4,4a,5,6,10b-hexah...)
Affinity DataIC50:  40nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313436(1-((2R,4aS,5R,10bS)-5-(4-fluorophenyl)-9-(trifluor...)
Affinity DataIC50:  58nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313433(CHEMBL1084431 | N-(2-aminoethyl)-4-methyl-N-(((2R,...)
Affinity DataIC50:  65nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340266(7-(2-(3-(4-chloro-2-methoxy-5-(trifluoromethyl)phe...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313401((4aS,5R,10bS)-7-fluoro-5-phenyl-9-(trifluoromethyl...)
Affinity DataIC50:  90nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313408(4-((4aS,5R,10bS)-9-tert-butyl-3,4,4a,5,6,10b-hexah...)
Affinity DataIC50:  95nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313391((4aS,5R,10bS)-5-phenyl-9-(trifluoromethyl)-3,4,4a,...)
Affinity DataIC50:  110nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340264(7-(2-(3-(5-chloro-2-methoxy-4-methylphenyl)ureido)...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340262(7-(2-(3-(2-methoxy-5-(trifluoromethyl)phenyl)ureid...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313419((4aS,5R,10bS)-9-tert-butyl-5-(thiophen-3-yl)-3,4,4...)
Affinity DataIC50:  120nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313387((4aS,5R,10bS)-9-ethyl-5-phenyl-3,4,4a,5,6,10b-hexa...)
Affinity DataIC50:  130nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313389((4aS,5R,10bS)-9-isopropyl-5-phenyl-3,4,4a,5,6,10b-...)
Affinity DataIC50:  130nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340273(CHEMBL1760633 | N-(6-(2-(3-(4-chloro-3-(trifluorom...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340259(7-(2-(3-(4-chloro-3-(trifluoromethyl)phenyl)ureido...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313414((4aS,5R,10bS)-9-tert-butyl-5-(2-fluorophenyl)-3,4,...)
Affinity DataIC50:  170nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340270(CHEMBL1760630 | N-(6-(2-(3-(2-methoxy-5-(trifluoro...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340285(CHEMBL1760736 | N-(6-(2-(3-(2-(2-aminoethoxy)-4-ch...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340277(CHEMBL1760637 | N-(6-(2-(3-(5-chloro-2-methoxy-4-m...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340265(7-(2-(3-(4-chloro-2-methoxy-5-methylphenyl)ureido)...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340288(CHEMBL1760617 | N-methyl-7-(2-(3-(3-(trifluorometh...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340258(CHEMBL1760619 | N-methyl-7-(2-(3-(4-methyl-3-(trif...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340281(CHEMBL1760641 | N-(6-(2-(3-(2-(2-(methylamino)etho...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340290(CHEMBL1760737 | N-(6-(2-(3-(2-(pyrrolidin-2-ylmeth...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340282(CHEMBL1760642 | N-(6-(2-(3-(4-chloro-2-(2-(methyla...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340260(7-(2-(3-(4-fluoro-3-(trifluoromethyl)phenyl)ureido...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340284(CHEMBL1760735 | N-(6-(2-(3-(2-(2-aminoethoxy)-5-(t...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50340261(7-(2-(3-(2-fluoro-5-(trifluoromethyl)phenyl)ureido...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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