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Found 60 with Last Name = 'antus' and Initial = 's'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347558(CHEMBL1802233)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347560(CHEMBL1802235)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataKi:  11.5nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347557(CHEMBL1802232)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347562(CHEMBL1802237)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347557(CHEMBL1802232)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347561(CHEMBL1802236)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347556(CHEMBL1802231)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347560(CHEMBL1802235)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347561(CHEMBL1802236)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347562(CHEMBL1802237)
Affinity DataKi:  415nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347559(CHEMBL1802234)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347558(CHEMBL1802233)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347559(CHEMBL1802234)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347556(CHEMBL1802231)
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50211296((7R,8S,9S,10R)-8,9,10-trihydroxy-7-hydroxymethyl-6...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50211294((7R,8S,9S,10R)-8,9,10-trihydroxy-7-hydroxymethyl-2...)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50211289(5-[4-(6,7-dibromo-2,3-dihydrobenzo[1,4]dioxin-2-yl...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50211288(5-[4-(6,7-dibromo-2,3-dihydrobenzo[1,4]dioxin-2-yl...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50211286(5-[4-(6-bromo-2,3-dihydrobenzo[1,4]dioxin-2-ylmeth...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of liver glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304282(CHEMBL610629 | N-((2R,3R,4S,5S,6R)-3,4,5-trihydrox...)
Affinity DataKi:  8.50E+4nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b by cheng-prusoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304281((S)-N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydrox...)
Affinity DataKi:  1.20E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b by cheng-prusoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304280((R)-N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydrox...)
Affinity DataKi:  1.28E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b by cheng-prusoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304278(8-methoxy-N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(...)
Affinity DataKi:  2.32E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b by cheng-prusoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304277(CHEMBL611030 | N-((2R,3R,4S,5S,6R)-3,4,5-trihydrox...)
Affinity DataKi:  2.52E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b by cheng-prusoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304279(8-bromo-N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hy...)
Affinity DataKi:  2.68E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b by cheng-prusoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  440nMAssay Description:Inhibition of bovine brain tubulin assessed as rate of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of bovine brain tubulin assessed as extent of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055045(CHEMBL3323243)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of bovine brain tubulin assessed as rate of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055045(CHEMBL3323243)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as extent of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304282(CHEMBL610629 | N-((2R,3R,4S,5S,6R)-3,4,5-trihydrox...)
Affinity DataIC50:  1.25E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50424716(NOSCAPINE | Narcotine | Tusscapine)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as rate of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055046(CHEMBL3323245)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as rate of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055044(CHEMBL3323241)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as rate of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304281((S)-N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydrox...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304280((R)-N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydrox...)
Affinity DataIC50:  3.20E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055043(CHEMBL3323244)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as rate of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055042(CHEMBL3323242)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as extent of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055042(CHEMBL3323242)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as rate of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055043(CHEMBL3323244)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as extent of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055041(CHEMBL3323240)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as rate of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055046(CHEMBL3323245)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as extent of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055041(CHEMBL3323240)
Affinity DataIC50: >4.00E+5nMAssay Description:Displacement of [3H]colchicine from bovine brain tubulin assessed as rate of assembly after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055042(CHEMBL3323242)
Affinity DataIC50: >4.00E+5nMAssay Description:Displacement of [3H]colchicine from bovine brain tubulin assessed as rate of assembly after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055043(CHEMBL3323244)
Affinity DataIC50: >4.00E+5nMAssay Description:Displacement of [3H]colchicine from bovine brain tubulin assessed as rate of assembly after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50424716(NOSCAPINE | Narcotine | Tusscapine)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as extent of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055041(CHEMBL3323240)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as extent of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50055044(CHEMBL3323241)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of bovine brain tubulin assessed as extent of assembly preincubated for 15 mins by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50304278(8-methoxy-N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(...)
Affinity DataIC50:  5.80E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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