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Found 114 with Last Name = 'babkov' and Initial = 'da'
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  10nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490649(CHEMBL2337184)
Affinity DataKi:  260nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490644(CHEMBL2337195)
Affinity DataKi:  310nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490643(CHEMBL2337196)
Affinity DataKi:  310nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490669(CHEMBL2337192)
Affinity DataKi:  550nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490662(CHEMBL2337194)
Affinity DataKi:  670nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490668(CHEMBL2337189)
Affinity DataKi:  1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490648(CHEMBL2337186)
Affinity DataKi:  1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490646(CHEMBL2337190)
Affinity DataKi:  1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063002(CHEMBL3398101)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490660(CHEMBL2337187)
Affinity DataKi:  6.50E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490642(CHEMBL2337197)
Affinity DataKi:  6.60E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490665(CHEMBL2337181)
Affinity DataKi:  6.60E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  7.20E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490659(CHEMBL2337174)
Affinity DataKi:  8.10E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490650(CHEMBL2337183)
Affinity DataKi:  1.00E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490647(CHEMBL2337188)
Affinity DataKi:  1.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490645(CHEMBL2337193)
Affinity DataKi:  1.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490653(CHEMBL2337173)
Affinity DataKi:  1.50E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063002(CHEMBL3398101)
Affinity DataKi:  1.54E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063002(CHEMBL3398101)
Affinity DataKi:  1.59E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063002(CHEMBL3398101)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490658(CHEMBL2337175)
Affinity DataKi:  2.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490663(CHEMBL2337191)
Affinity DataKi:  2.90E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490657(CHEMBL2337182)
Affinity DataKi:  4.70E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490652(CHEMBL2337177)
Affinity DataKi:  5.10E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490654(CHEMBL2337201)
Affinity DataKi:  5.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063002(CHEMBL3398101)
Affinity DataKi:  6.33E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063002(CHEMBL3398101)
Affinity DataKi:  6.76E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490656(CHEMBL2337198)
Affinity DataKi:  6.80E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063002(CHEMBL3398101)
Affinity DataKi:  6.99E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490661(CHEMBL2337176)
Affinity DataKi:  7.10E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063001(CHEMBL3398091)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063003(CHEMBL3398092)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063013(CHEMBL3398083)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063014(CHEMBL3398084)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063010(CHEMBL3398082)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063017(CHEMBL3398085)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063018(CHEMBL3398086)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063019(CHEMBL3398087)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063020(CHEMBL3398088)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063022(CHEMBL3398089)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50063023(CHEMBL3398090)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490651(CHEMBL2337179)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490655(CHEMBL2337199)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490664(CHEMBL2337185)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490666(CHEMBL2337178)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490667(CHEMBL2337200)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490670(CHEMBL2337180)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Lomonosov Moscow State University

Curated by ChEMBL
LigandPNGBDBM50523811(CHEMBL2094331 | DNDI1416941)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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