TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 670nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.50E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.60E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.60E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 7.20E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 8.10E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.54E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.59E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 2.90E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 4.70E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 5.10E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 5.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.33E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.76E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.80E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.99E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 7.10E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair