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Found 48 with Last Name = 'bacalhau' and Initial = 'p'
TargetCholinesterase(Equus caballus (Horse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataKi:  4.10E+4nMAssay Description:Reversible competitive inhibition of equine BuChE by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50344826(1-(4-chlorobenzyl)-3-hydroxy-3-phenylindolin-2-one...)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of AChE in Swiss mouse brain homogenate using acetylthiocholine iodide as substrate by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  3.50E+3nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503820(CHEMBL4550082)
Affinity DataIC50:  6.61E+3nMAssay Description:Inhibition of equine serum BuChE after 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503818(CHEMBL4593576)
Affinity DataIC50:  7.41E+3nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  6.19E+4nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM192007(Isoquinolin-1(2H)-ones, 1f)
Affinity DataIC50:  8.95E+4nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM191998(Isoquinolin-1(2H)-ones, 2b)
Affinity DataIC50:  1.08E+5nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM191997(Isoquinolin-1(2H)-ones, 2a)
Affinity DataIC50:  1.08E+5nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM192000(Isoquinolin-1(2H)-ones, 2d)
Affinity DataIC50:  1.09E+5nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  1.25E+5nMAssay Description:Inhibition of AChE in Swiss mouse liver homogenate using acetylthiocholine iodide as substrate by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM50344826(1-(4-chlorobenzyl)-3-hydroxy-3-phenylindolin-2-one...)
Affinity DataIC50:  1.29E+5nMAssay Description:Inhibition of electrophorus electricus AChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM191992(Isoquinolin-1(2H)-ones, 1a)
Affinity DataIC50:  1.36E+5nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  1.47E+5nMAssay Description:Inhibition of BuChE in Swiss mouse liver homogenate by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM192007(Isoquinolin-1(2H)-ones, 1f)
Affinity DataIC50:  1.54E+5nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM50503820(CHEMBL4550082)
Affinity DataIC50:  1.93E+5nMAssay Description:Inhibition of electrophorus electricus AChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM191995(Isoquinolin-1(2H)-ones, 1d)
Affinity DataIC50:  2.26E+5nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM50503818(CHEMBL4593576)
Affinity DataIC50:  2.37E+5nMAssay Description:Inhibition of electrophorus electricus AChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM191999(Isoquinolin-1(2H)-ones, 2c)
Affinity DataIC50:  2.69E+5nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM191997(Isoquinolin-1(2H)-ones, 2a)
Affinity DataIC50:  2.78E+5nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM191996(Isoquinolin-1(2H)-ones, 1e)
Affinity DataIC50:  3.11E+5nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM191993(Isoquinolin-1(2H)-ones, 1b)
Affinity DataIC50:  3.52E+5nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataIC50:  4.35E+5nMAssay Description:Inhibition of BuChE in Swiss mouse liver homogenate by Ellman's assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of electrophorus electricus AChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM191998(Isoquinolin-1(2H)-ones, 2b)
Affinity DataIC50:  5.36E+5nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM192003(Isoquinolin-1(2H)-ones, 4a)
Affinity DataIC50:  5.50E+5nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM191999(Isoquinolin-1(2H)-ones, 2c)
Affinity DataIC50:  5.64E+5nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataIC50:  5.65E+5nMAssay Description:Inhibition of AChE in Swiss mouse liver homogenate using acetylthiocholine iodide as substrate by Ellman's assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM192000(Isoquinolin-1(2H)-ones, 2d)
Affinity DataIC50:  5.85E+5nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM192006(Isoquinolin-1(2H)-ones, 6)
Affinity DataIC50:  7.56E+5nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM191992(Isoquinolin-1(2H)-ones, 1a)
Affinity DataIC50:  8.08E+5nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM192006(Isoquinolin-1(2H)-ones, 6)
Affinity DataIC50:  8.26E+5nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM192002(Isoquinolin-1(2H)-ones, 3b)
Affinity DataIC50:  1.25E+6nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM192001(Isoquinolin-1(2H)-ones, 3a)
Affinity DataIC50:  1.30E+6nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM192005(Isoquinolin-1(2H)-ones, 5)
Affinity DataIC50:  1.37E+6nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM191993(Isoquinolin-1(2H)-ones, 1b)
Affinity DataIC50: >1.50E+6nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM191994(Isoquinolin-1(2H)-ones, 1c)
Affinity DataIC50: >1.50E+6nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM191995(Isoquinolin-1(2H)-ones, 1d)
Affinity DataIC50: >1.50E+6nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM191996(Isoquinolin-1(2H)-ones, 1e)
Affinity DataIC50: >1.50E+6nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM192005(Isoquinolin-1(2H)-ones, 5)
Affinity DataIC50: >1.50E+6nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM192004(Isoquinolin-1(2H)-ones, 4b)
Affinity DataIC50: >1.50E+6nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM192003(Isoquinolin-1(2H)-ones, 4a)
Affinity DataIC50: >1.50E+6nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM192002(Isoquinolin-1(2H)-ones, 3b)
Affinity DataIC50: >1.50E+6nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM192001(Isoquinolin-1(2H)-ones, 3a)
Affinity DataIC50: >1.50E+6nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universidade De Evora

LigandPNGBDBM191994(Isoquinolin-1(2H)-ones, 1c)
Affinity DataIC50: >1.50E+6nMAssay Description:The in vitro BuChE assay was performed similarly to the method described above. A standard enzyme activity curve was drawn for each enzyme using seve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade De Evora

LigandPNGBDBM192004(Isoquinolin-1(2H)-ones, 4b)
Affinity DataIC50: >1.50E+6nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed