TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 48.5nMAssay Description:Inhibition of mushroom tyrosinase by kinetic based assayMore data for this Ligand-Target Pair
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 181nMAssay Description:Inhibition of mushroom tyrosinase by kinetic based assayMore data for this Ligand-Target Pair
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Inhibition of monophenolase activity of mushroom tyrosinase using as L-tyrosine substrate by Lineweaver-Burk plot based kinetic assayMore data for this Ligand-Target Pair
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using as L-DOPA substrate by Lineweaver-Burk plot based kinetic assayMore data for this Ligand-Target Pair
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Affinity DataKi: 350nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Inhibition of monophenolase activity of mushroom tyrosinase using as L-tyrosine substrate by Lineweaver-Burk plot based kinetic assayMore data for this Ligand-Target Pair
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 770nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using as L-DOPA substrate by Lineweaver-Burk plot based kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 870nMAssay Description:Inhibition of mushroom tyrosinase by kinetic based assayMore data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Pohang University Of Science And Technology
Curated by PDSP Ki Database
Affinity DataKi: 1.45E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.33E+3nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.36E+3nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.39E+3nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.63E+3nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.12E+3nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nM ΔG°: -31.9kJ/mole IC50: 1.02E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataKi: 4.39E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.35E+3nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.58E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.63E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.83E+3nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.39E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.65E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.04E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.40E+3nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 9.12E+3nMAssay Description:Inhibition of monophenolase activity of mushroom tyrosinase using as L-tyrosine substrate by Lineweaver-Burk plot based kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.31E+3nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 1.08E+4nMAssay Description:Inhibition of monophenolase activity of mushroom tyrosinase using as L-tyrosine substrate by Lineweaver-Burk plot based kinetic assayMore data for this Ligand-Target Pair
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 1.12E+4nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using as L-DOPA substrate by Lineweaver-Burk plot based kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.23E+4nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.31E+4nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 1.56E+4nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using as L-DOPA substrate by Lineweaver-Burk plot based kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Inhibition of human NOX4 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Inhibition of human NOX1 expressed in Drosophila DUOX knockdown model assessed as decrease in ROS production by lucigenin chemiluminescence assayMore data for this Ligand-Target Pair