Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]-PDBU from protein kinase C-alphaMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]-PDBU from protein kinase C-alphaMore data for this Ligand-Target Pair
Affinity DataKi: 165nMAssay Description:Displacement of [3H]-PDBU from protein kinase C-alphaMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase C (alpha)More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Displacement of [3H]-PDBU from protein kinase C-alphaMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase C (alpha)More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase C (alpha)More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase C (alpha)More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair