Compile Data Set for Download or QSAR
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Found 594 with Last Name = 'barnett' and Initial = 'sf'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243218(2-(4-((4-(5-(6-oxo-1,6-dihydropyridin-3-yl)-4H-1,2...)
Affinity DataIC50:  1nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256715(9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-triaz...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256714(9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-triaz...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256723(9-phenyl-8-(4-((4-(4-(pyridin-2-yl)-1H-imidazol-1-...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243221(2-(4-((4-(5-(6-methoxypyridin-3-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256723(9-phenyl-8-(4-((4-(4-(pyridin-2-yl)-1H-imidazol-1-...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243215(3-phenyl-2-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256713(3-phenyl-2-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-triaz...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24876(2-{5-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3...)
Affinity DataIC50:  3.80nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243220(3-phenyl-2-(4-((4-(5-(pyrazin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256718(9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-triaz...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243219(2-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-triazol...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24883(1-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]...)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24875(4-{3-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3...)
Affinity DataIC50:  4.5nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256719(3-methyl-9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243776(2-(1H-imidazol-1-yl)-6-phenyl-7-(4-((4-(5-(pyridin...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243777(1-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256718(9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-triaz...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Akt1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243764(2-morpholino-6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50373461(CHEMBL259753)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24880(CHEMBL252857 | N-methyl-6-phenyl-7-[4-({4-[5-(pyri...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24880(CHEMBL252857 | N-methyl-6-phenyl-7-[4-({4-[5-(pyri...)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24879(6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  6.20nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256715(9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-triaz...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243778(2-(4-(methylsulfonyl)piperazin-1-yl)-6-phenyl-7-(4...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243217(3-phenyl-2-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2,4-tri...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243765(1-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-tr...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50373462(CHEMBL259967)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243769(2-((R)-3-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243218(2-(4-((4-(5-(6-oxo-1,6-dihydropyridin-3-yl)-4H-1,2...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24872(5-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]...)
Affinity DataIC50:  8.5nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256717(1-(9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-tr...)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243771(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243782(2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256714(9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-triaz...)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24873(1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyr...)
Affinity DataIC50:  9.70nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256721(3-((4-methylpiperazin-1-yl)methyl)-9-phenyl-8-(4-(...)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243775(CHEMBL454859 | N,N-dimethyl-1-(6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256718(9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-triaz...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243286(CHEMBL499554 | N,N-dimethyl-2-(4-(2-phenyl-3-(4-((...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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