Compile Data Set for Download or QSAR
maximum 50k data
Found 20 with Last Name = 'bartlett' and Initial = 'rd'
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50366944(Azovan Blue | Azovan sodium | EVANS BLUE)
Affinity DataKi:  40nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113317(Bis[4-Amino-5-hydroxy-6-(2-methoxy-phenylazo)-naph...)
Affinity DataKi:  190nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50089912((2S)-2-amino-4-methylidenepentanedioic acid | 4-me...)
Affinity DataKi:  3.00E+3nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113314(6-Biphenyl-4-yl-quinoline-2,4-dicarboxylic acid | ...)
Affinity DataKi:  4.10E+4nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113320(6-(2-Biphenyl-4-yl-vinyl)-quinoline-2,4-dicarboxyl...)
Affinity DataKi:  6.40E+4nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113314(6-Biphenyl-4-yl-quinoline-2,4-dicarboxylic acid | ...)
Affinity DataKi:  9.50E+4nMAssay Description:Inhibitory conc. against Vesicular glutamate transporter (VGLUT), derived from Lineweaver-Burke analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113318(6-Styryl-quinoline-2,4-dicarboxylic acid | CHEMBL7...)
Affinity DataKi:  1.29E+5nMAssay Description:Inhibitory conc. against Vesicular glutamate transporter (VGLUT), derived from Lineweaver-Burke analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113321(6-Phenethyl-quinoline-2,4-dicarboxylic acid | CHEM...)
Affinity DataKi:  1.43E+5nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113318(6-Styryl-quinoline-2,4-dicarboxylic acid | CHEMBL7...)
Affinity DataKi:  1.67E+5nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113323(6-Phenethyloxy-quinoline-2,4-dicarboxylic acid | C...)
Affinity DataKi:  1.89E+5nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113313(4,8-Dihydroxy-quinoline-2-carboxylic acid anion | ...)
Affinity DataKi:  1.90E+5nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent phosphate transport protein 1(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50081123(6-Benzyloxy-quinoline-2,4-dicarboxylic acid | CHEM...)
Affinity DataKi:  2.04E+5nMAssay Description:Compound was evaluated for the binding affinity against glutamate vesicular transport (GVT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50081123(6-Benzyloxy-quinoline-2,4-dicarboxylic acid | CHEM...)
Affinity DataKi:  2.04E+5nMAssay Description:Inhibitory conc. against Vesicular glutamate transporter (VGLUT), derived from Lineweaver-Burke analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113319(8-Hydroxy-quinoline-2,4-dicarboxylic acid | CHEMBL...)
Affinity DataKi:  2.86E+5nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113322(6-Phenylazo-quinoline-2,4-dicarboxylic acid | CHEM...)
Affinity DataKi:  2.88E+5nMAssay Description:Compound was evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported,.using Cheng-Prushoff eq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50081123(6-Benzyloxy-quinoline-2,4-dicarboxylic acid | CHEM...)
Affinity DataKi:  3.68E+5nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50005001(7-Chloro-4-hydroxy-quinoline-2-carboxylic acid | 7...)
Affinity DataKi:  5.90E+5nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50060136((1R,3S)-1-Amino-cyclopentane-1,3-dicarboxylic acid...)
Affinity DataKi:  7.00E+5nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM81975(4-hydroxyquinoline-2-carboxylic acid | CAS_492-27-...)
Affinity DataKi:  1.30E+6nMAssay Description:Compound was evaluated for the inhibition of Vesicular glutamate transporter (VGLUT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113315(5-Bromo-7-methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3...)
Affinity DataIC50:  2.20E+4nMAssay Description:Compound was evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed