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Found 219 with Last Name = 'batchelor' and Initial = 'm'
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Celltech Therapeutics

Curated by ChEMBL
LigandPNGBDBM50083639(CHEMBL112346 | {4-[6-((S)-3-Ethyl-piperazin-1-yl)-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Zeta-chain (TCR) associated protein kinase 70 kDa phosphorylation of polyGly-Tyr.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295759(1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)-6-(...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295752(4-(6-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)-1H-pyrro...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295760(1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)-1H-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295754((4-(1-(benzo[c][1,2,5]oxadiazol-4-ylsulfonyl)-1H-p...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Celltech Therapeutics

Curated by ChEMBL
LigandPNGBDBM50083638((S)-4-(6-(3-methylpiperazin-1-yl)pyridin-3-yl)-N-(...)
Affinity DataIC50:  11nMAssay Description:Inhibition of Zeta-chain (TCR) associated protein kinase 70 kDa phosphorylation of polyGly-Tyr.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295755(1-(4-(1-(benzo[c][1,2,5]oxadiazol-4-ylsulfonyl)-1H...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295756(1-(4-(1-(benzo[c][1,2,5]oxadiazol-4-ylsulfonyl)-1H...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295750(4-(6-(6-(4-methylpiperazin-1-yl)pyridin-3-yl)-1H-p...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295761(1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)-1H-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295753(1-(benzo[c][1,2,5]oxadiazol-4-ylsulfonyl)-1H-pyrro...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50265989(CHEMBL462707 | N-(3-(4-methylpiperazin-1-yl)-7-(tr...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant his-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262463((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-7,7-di...)
Affinity DataIC50:  18nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295767(4-((6-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)-1H-pyrr...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295764(1-benzyl-1H-pyrrolo[3,2-b]pyridine | CHEMBL561256)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295763(CHEMBL564440 | tert-butyl 4-(4-(1-(6-chloroimidazo...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295748(1-(2-nitrophenylsulfonyl)-6-(piperazin-1-yl)-1H-py...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295747(CHEMBL556627 | tert-butyl 4-(1-(2-nitrophenylsulfo...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295735(1-(2-nitrophenylsulfonyl)-1H-pyrrolo[3,2-b]pyridin...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295749(4-(1H-pyrrolo[3,2-b]pyridin-1-ylsulfonyl)benzo[c][...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295751(4-(6-(piperazin-1-yl)-1H-pyrrolo[3,2-b]pyridin-1-y...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295758(1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)-6-(...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Celltech Therapeutics

Curated by ChEMBL
LigandPNGBDBM50083649(CHEMBL112518 | {4-[6-(3-Methyl-piperazin-1-yl)-pyr...)
Affinity DataIC50:  26nMAssay Description:Inhibition of Zeta-chain (TCR) associated protein kinase 70 kDa phosphorylation of polyGly-Tyr.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295762(CHEMBL550158 | tert-butyl 4-(1-(6-chloroimidazo[2,...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Celltech Therapeutics

Curated by ChEMBL
LigandPNGBDBM50083640(CHEMBL112172 | [4-(6-[1,4]Diazepan-1-yl-pyridin-3-...)
Affinity DataIC50:  31nMAssay Description:Inhibition of Zeta-chain (TCR) associated protein kinase 70 kDa phosphorylation of polyGly-Tyr.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50266023(CHEMBL515659 | N-(benzo[c][1,2,5]oxadiazol-4-ylmet...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human recombinant his-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262463((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-7,7-di...)
Affinity DataIC50:  31nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295769(CHEMBL564827 | tert-butyl 4-(4-(1-(benzo[c][1,2,5]...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295757(1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)-1H-...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262460((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  35nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50265954(3-(4-methylpiperazin-1-yl)-N-(3-nitrobenzyl)-7-(tr...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant his-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Celltech Therapeutics

Curated by ChEMBL
LigandPNGBDBM50083648(CHEMBL420672 | {4-[6-(4-Methyl-piperazin-1-yl)-pyr...)
Affinity DataIC50:  46nMAssay Description:Inhibition of Zeta-chain (TCR) associated protein kinase 70 kDa phosphorylation of polyGly-Tyr.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262460((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  49nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262460((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  51nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Celltech Therapeutics

Curated by ChEMBL
LigandPNGBDBM50083644(CHEMBL322066 | [4-(6-Piperazin-1-yl-pyridin-3-yl)-...)
Affinity DataIC50:  54nMAssay Description:Inhibition of Zeta-chain (TCR) associated protein kinase 70 kDa phosphorylation of polyGly-Tyr.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50265987(3-(4-methylpiperazin-1-yl)-N-(4-nitrobenzyl)-7-(tr...)
Affinity DataIC50:  55nMAssay Description:Inhibition of human recombinant his-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262463((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-7,7-di...)
Affinity DataIC50:  59nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262462((S)-2-(3-(benzo[b]thiophen-3-ylmethyl)morpholino)-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262461(2-(3-((1H-pyrrolo[2,3-b]pyridin-3-yl)methyl)morpho...)
Affinity DataIC50:  63nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295734(1-(3-nitrophenylsulfonyl)-1H-pyrrolo[3,2-b]pyridin...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262461(2-(3-((1H-pyrrolo[2,3-b]pyridin-3-yl)methyl)morpho...)
Affinity DataIC50:  74nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295742(3-(2-nitrophenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin...)
Affinity DataIC50:  75nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295745(1-(2-nitrophenylsulfonyl)-1H-pyrrolo[3,2-b]pyridin...)
Affinity DataIC50:  82nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295759(1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)-6-(...)
Affinity DataIC50:  90nMAssay Description:Inhibition of c-Met phosphorylation in human A549 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295731(1-(2,3-dichlorophenylsulfonyl)-1H-pyrrolo[3,2-b]py...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant His-tagged c-Met by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262461(2-(3-((1H-pyrrolo[2,3-b]pyridin-3-yl)methyl)morpho...)
Affinity DataIC50:  107nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295759(1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)-6-(...)
Affinity DataIC50:  110nMAssay Description:Inhibition of c-Met phosphorylation in human MKN45 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50295762(CHEMBL550158 | tert-butyl 4-(1-(6-chloroimidazo[2,...)
Affinity DataIC50:  110nMAssay Description:Inhibition of c-Met phosphorylation in human A549 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262462((S)-2-(3-(benzo[b]thiophen-3-ylmethyl)morpholino)-...)
Affinity DataIC50:  125nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Celltech Therapeutics

Curated by ChEMBL
LigandPNGBDBM50083641(Aminopyrimidine (Scaffold II) | CHEMBL113185 | N*1...)
Affinity DataIC50:  125nMAssay Description:Inhibition of Zeta-chain (TCR) associated protein kinase 70 kDa phosphorylation of polyGly-Tyr.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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