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Found 214 with Last Name = 'bobkova' and Initial = 'e'
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM88776(2-[4-[(Z)-[5-(4-chlorophenyl)-6-isopropoxycarbonyl...)
Affinity DataKi:  690nMAssay Description:Competitive inhibition of recombinant HePTP expressed in Escherichia coli by Michaelis-Menten kinetic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447413(CHEMBL3115157)
Affinity DataKi:  3.20E+3nMAssay Description:Competitive inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells using p-nitrophenyl phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM92490(Compound # 1)
Affinity DataIC50:  11nMAssay Description:1536-Well TR-Fret uHTS assay PDK1-tide1 peptide substrate.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM92490(Compound # 1)
Affinity DataIC50:  14nMAssay Description:384-Well TR-Fret assay using AKT-tide peptide substrate.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM26198(4-tert-butyl-15-fluoro-3,5,10-triazatetracyclo[11....)
Affinity DataIC50:  20nMAssay Description:1536-Well TR-Fret uHTS assay PDK1-tide1 peptide substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM26198(4-tert-butyl-15-fluoro-3,5,10-triazatetracyclo[11....)
Affinity DataIC50:  28nMAssay Description:384-Well TR-Fret assay using AKT-tide peptide substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM76214(CHEMBL1322977 | MLS001096094 | N-(2,5-dimethylphen...)
Affinity DataIC50:  400nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM47952(MLS000588669 | N-(1-allyl-3-tosyl-pyrrolo[3,2-b]qu...)
Affinity DataIC50:  500nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM54915(MLS000588658 | N-(1-butyl-3-tosyl-pyrrolo[3,2-b]qu...)
Affinity DataIC50:  500nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447450(CHEMBL3115119)
Affinity DataIC50:  530nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447413(CHEMBL3115157)
Affinity DataIC50:  540nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447458(CHEMBL3115158)
Affinity DataIC50:  730nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM30831(MLS000055622 | N-(1-butyl-3-cyano-2-pyrrolo[3,2-b]...)
Affinity DataIC50:  760nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM88776(2-[4-[(Z)-[5-(4-chlorophenyl)-6-isopropoxycarbonyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM160656(US9045483, 9)
Affinity DataIC50:  1.10E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50378898(CHEMBL1672292)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447426(CHEMBL3115137)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447415(CHEMBL3115148)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50378899(CHEMBL1672293)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM76215(CHEMBL1349252 | MLS001096095 | N-(3-cyanophenyl)-3...)
Affinity DataIC50:  1.82E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447449(CHEMBL3115120)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447425(CHEMBL3115138)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447457(CHEMBL3115159)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447448(CHEMBL3115121)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447447(CHEMBL3115122)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM32062(MLS000054842 | N-(1-butyl-3-cyano-2-pyrrolo[3,2-b]...)
Affinity DataIC50:  3.60E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50336847(2-(4-((5-(2-chlorophenyl)-6-(ethoxycarbonyl)-7-met...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447413(CHEMBL3115157)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells using p-nitrophenyl phosphate as substrate after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447424(CHEMBL3115139)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50378898(CHEMBL1672292)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM160655(US9045483, 8)
Affinity DataIC50:  4.50E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50336848(2-(4-((6-(ethoxycarbonyl)-5-(3-methoxyphenyl)-7-me...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447456(CHEMBL3115160)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM92492(Alkaloid 1)
Affinity DataIC50:  5.70E+3nMAssay Description:1536-Well TR-Fret uHTS assay PDK1-tide1 peptide substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM160657(US9045483, 10)
Affinity DataIC50:  5.70E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447422(CHEMBL3115141)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50336847(2-(4-((5-(2-chlorophenyl)-6-(ethoxycarbonyl)-7-met...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447423(CHEMBL3115140)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447446(CHEMBL3115123)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM37640(MLS000079917 | N-(1-butyl-3-cyano-2-pyrrolo[3,2-b]...)
Affinity DataIC50:  8.30E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50378899(CHEMBL1672293)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50336848(2-(4-((6-(ethoxycarbonyl)-5-(3-methoxyphenyl)-7-me...)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447445(CHEMBL3115124)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447421(CHEMBL3115142)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM92493(Alkaloid 2)
Affinity DataIC50:  1.80E+4nMAssay Description:1536-Well TR-Fret uHTS assay PDK1-tide1 peptide substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447443(CHEMBL3115125)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM88776(2-[4-[(Z)-[5-(4-chlorophenyl)-6-isopropoxycarbonyl...)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM30722(MLS000068755 | N-(1-butyl-3-cyano-2-pyrrolo[3,2-b]...)
Affinity DataIC50:  2.00E+4nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAlkaline phosphatase, germ cell type(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447413(CHEMBL3115157)
Affinity DataIC50:  2.11E+4nMAssay Description:Inhibition of mouse EAP using p-nitrophenyl phosphate as substrate after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1/2(Homo sapiens (Human))
City Of Hope

US Patent
LigandPNGBDBM43094(2-chloranyl-N-[3-cyano-1-(phenylmethyl)pyrrolo[3,2...)
Affinity DataIC50:  2.50E+4nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In DepthDetails US Patent
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