TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 148nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 166nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 263nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 269nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 269nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 309nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 339nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 398nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 501nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 525nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 537nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cell membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 398nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 372nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 63nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 5.01E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 155nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 2.88E+3nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 2.51E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 62nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 3.16E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair