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Found 53 with Last Name = 'camacho gomez' and Initial = 'ja'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128311(US8796284, 93)
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128297(US8796284, 4)
Affinity DataKi:  6nM ΔG°:  -46.9kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128310(US8796284, 48)
Affinity DataKi:  7nM ΔG°:  -46.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128307(US8796284, 38)
Affinity DataKi:  7nM ΔG°:  -46.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128306(US8796284, 36)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128305(US8796284, 29)
Affinity DataKi:  10nM ΔG°:  -45.7kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128296(US8796284, 3)
Affinity DataKi:  11nM ΔG°:  -45.4kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128295(US8796284, 1)
Affinity DataKi:  12nM ΔG°:  -45.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128311(US8796284, 93)
Affinity DataKi:  12nM ΔG°:  -47.0kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128308(US8796284, 44)
Affinity DataKi:  14nM ΔG°:  -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128303(US8796284, 20)
Affinity DataKi:  14nM ΔG°:  -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128298(US8796284, 5)
Affinity DataKi:  14nM ΔG°:  -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128304(US8796284, 24)
Affinity DataKi:  16nM ΔG°:  -44.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128309(US8796284, 46)
Affinity DataKi:  17nM ΔG°:  -44.3kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128299(US8796284, 8)
Affinity DataKi:  18nM ΔG°:  -44.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128301(US8796284, 10)
Affinity DataKi:  21nM ΔG°:  -43.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128295(US8796284, 1)
Affinity DataKi:  25nM ΔG°:  -45.1kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128300(US8796284, 9)
Affinity DataKi:  33nM ΔG°:  -42.7kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128302(US8796284, 13)
Affinity DataKi:  35nM ΔG°:  -42.6kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128302(US8796284, 13)
Affinity DataKi:  50nM ΔG°:  -43.3kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM128299(US8796284, 8)
Affinity DataKi:  60nM ΔG°:  -42.9kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474288(CHEMBL112192)
Affinity DataIC50:  220nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474300(CHEMBL116173)
Affinity DataIC50:  370nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on TubulinMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474288(CHEMBL112192)
Affinity DataIC50:  430nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474290(CHEMBL115499)
Affinity DataIC50:  480nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474293(CHEMBL324797)
Affinity DataIC50:  630nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474298(CHEMBL321632)
Affinity DataIC50:  630nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474300(CHEMBL116173)
Affinity DataIC50:  670nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474308(CHEMBL112385)
Affinity DataIC50:  760nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM97233(CHEMBL9514 | MLS001164242 | N-[6-(2-thenoyl)-1H-be...)
Affinity DataIC50:  760nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474286(CHEMBL419387)
Affinity DataIC50:  910nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474287(CHEMBL115488)
Affinity DataIC50:  910nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50469124(CHEMBL113332)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  1.26E+3nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on tubulinMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474291(CHEMBL326388)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474294(CHEMBL115360)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474292(CHEMBL114642)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474307(CHEMBL114651)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474306(CHEMBL326114)
Affinity DataIC50:  2.60E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474299(CHEMBL267340)
Affinity DataIC50:  4.40E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474302(CHEMBL327061)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474289(CHEMBL326395)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474304(CHEMBL114937)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474305(CHEMBL422965)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474285(CHEMBL115490)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474295(CHEMBL114677)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474301(CHEMBL114423)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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