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Found 31 with Last Name = 'cambareri' and Initial = 'a'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092516(3-{[(Methoxycarbonyl-pyridin-2-yl-methyl)-methyl-a...)
Affinity DataKi:  15nMAssay Description:Inhibition against [3H]-CI 977 rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092518(3-[{[Methoxycarbonyl-(4-methoxy-phenyl)-methyl]-me...)
Affinity DataKi:  18nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1 at 10 micromol/LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092515(3-((3-Hydroxy-phenyl)-{[(3-hydroxy-phenyl)-methoxy...)
Affinity DataKi:  20nMAssay Description:Inhibition against [3H]-CI 977 rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092521(3-((3-Fluoro-phenyl)-{[(3-fluoro-phenyl)-methoxyca...)
Affinity DataKi:  26nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092520(3-((4-Fluoro-phenyl)-{[(4-fluoro-phenyl)-methoxyca...)
Affinity DataKi:  140nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1 at 10 micromol/LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092519(3-{[(Methoxycarbonyl-quinolin-2-yl-methyl)-methyl-...)
Affinity DataKi:  190nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092517(3-{[(Carboxy-phenyl-methyl)-methyl-amino]-phenyl-m...)
Affinity DataKi:  210nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1 at 10 micromol/LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092514(3-{[(Methoxycarbonyl-m-tolyl-methyl)-methyl-amino]...)
Affinity DataKi:  820nMAssay Description:Inhibition against [3H]-CI 977 rat Opioid receptor kappa 1 at 10 micromol/LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092513(3-((4-Chloro-phenyl)-{[(4-chloro-phenyl)-ethoxycar...)
Affinity DataKi:  1.98E+3nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074561(Bis-{4-{[3-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-p...)
Affinity DataEC50:  5.08E+4nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074563(Bis-{4-[(1,3-Dioxo-1,3-dihydro-isoindol-2-ylmethox...)
Affinity DataEC50:  1.40E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074565(2-{2-[4-(3-{1-[2-(1,3-dioxo-2,3-dihydro-1H-2-isoin...)
Affinity DataEC50:  4.87E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074564(Bis-{3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  2.69E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074566(2-{4-[4-(3-{1-[4-(1,3-dioxo-2,3-dihydro-1H-2-isoin...)
Affinity DataEC50:  4.65E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074568(Bis-{4-{[3-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-p...)
Affinity DataEC50:  350nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074567(Bis-{4-{[3-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-p...)
Affinity DataEC50:  510nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074569((6-{bis[3-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-pr...)
Affinity DataEC50:  1.44E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074570(2-(4-{3-[1-(1,3-dioxo-2,3-dihydro-1H-2-isoindolylm...)
Affinity DataEC50:  3.49E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074571(Bis-{4-{[3-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-p...)
Affinity DataEC50:  450nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074573(Bis-{3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  570nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074572(2-{3-[4-(3-{1-[3-(1,3-dioxo-2,3-dihydro-1H-2-isoin...)
Affinity DataEC50:  630nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074562(Bis-{4-[(1,3-Dioxo-1,3-dihydro-isoindol-2-ylmethox...)
Affinity DataEC50:  1.90E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074558(Bis-{3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  370nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074559(Bis-[3-(1,3-dioxo-1,3-dihydro-isoindol-2-yl)-propy...)
Affinity DataEC50:  8.82E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074560(Bis-{3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  530nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074557(Bis-{4-{[3-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-p...)
Affinity DataEC50:  520nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074556(Bis-{4-[(1,3-Dioxo-1,3-dihydro-isoindol-2-ylmethox...)
Affinity DataEC50:  510nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074555(Bis-{3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  1.39E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074554(2-[4-(4-{1-[4-(1,3-dioxo-2,3-dihydro-1H-2-isoindol...)
Affinity DataEC50:  470nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074552(Bis-[3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  3.80E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50074553(2-{4-[4-(2-{1-[4-(1,3-dioxo-2,3-dihydro-1H-2-isoin...)
Affinity DataEC50:  2.34E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]-N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed