TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Sosei Heptares
Curated by ChEMBL
Sosei Heptares
Curated by ChEMBL
Affinity DataKi: 0.0200nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Sosei Heptares
Curated by ChEMBL
Sosei Heptares
Curated by ChEMBL
Affinity DataKi: 0.0251nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Sosei Heptares
Curated by ChEMBL
Sosei Heptares
Curated by ChEMBL
Affinity DataKi: 0.0316nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Sosei Heptares
Curated by ChEMBL
Sosei Heptares
Curated by ChEMBL
Affinity DataKi: 0.0316nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Sosei Heptares
Curated by ChEMBL
Sosei Heptares
Curated by ChEMBL
Affinity DataKi: 0.0398nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Sosei Heptares
Curated by ChEMBL
Sosei Heptares
Curated by ChEMBL
Affinity DataKi: 0.0631nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Sosei Heptares
Curated by ChEMBL
Sosei Heptares
Curated by ChEMBL
Affinity DataKi: 0.0794nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Sosei Heptares
Curated by ChEMBL
Sosei Heptares
Curated by ChEMBL
Affinity DataKi: 0.0794nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Sosei Heptares
Curated by ChEMBL
Sosei Heptares
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintill...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.660nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.930nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 6nM EC50: 40nMAssay Description:The assay is based upon displacement of a fluorescently labeled molecule, which binds specifically to the ATP-binding site of full-length human Hsp90...More data for this Ligand-Target Pair
Affinity DataIC50: 6nM EC50: 6nMAssay Description:The assay is based upon displacement of a fluorescently labeled molecule, which binds specifically to the ATP-binding site of full-length human Hsp90...More data for this Ligand-Target Pair