Compile Data Set for Download or QSAR
maximum 50k data
Found 31 with Last Name = 'caporuscio' and Initial = 'f'
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345657(CHEMBL1784801 | rac-3-((1H-imidazol-1-yl)methyl)-1...)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345645(CHEMBL1485809 | rac-1-(1H-imidazol-1-yl)-3-phenoxy...)
Affinity DataIC50:  16.5nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345671(CHEMBL1784811 | rac-1-(2-((1H-imidazol-1-yl)methyl...)
Affinity DataIC50:  34.5nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345672(CHEMBL1784812 | rac-1-(2-((1H-imidazol-1-yl)methyl...)
Affinity DataIC50:  46.7nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345648(CHEMBL1784791 | rac-1-(2-((1H-imidazol-1-yl)methyl...)
Affinity DataIC50:  59.2nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345665(CHEMBL1784807 | N-(3-(1H-imidazol-1-yl)propyl)-4-m...)
Affinity DataIC50:  61.6nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345666(CHEMBL1351273 | N-(3-(1H-imidazol-1-yl)propyl)-2,5...)
Affinity DataIC50:  63.7nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345660(CHEMBL1784805 | rac-1-(4-(2-((1H-imidazol-1-yl)met...)
Affinity DataIC50:  66.5nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345659(CHEMBL1784804 | rac-2-((1H-imidazol-1-yl)methyl)-4...)
Affinity DataIC50:  78.8nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345669(CHEMBL1784809 | N-(3-(1H-imidazol-1-yl)propyl)-3-f...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345646(CHEMBL1784789 | N-(3-(1H-imidazol-1-yl)propyl)-2,3...)
Affinity DataIC50:  119nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345664(CHEMBL1303900 | N-(3-(1H-imidazol-1-yl)propyl)-2,4...)
Affinity DataIC50:  172nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345655(CHEMBL1784798 | N-(2-(4-fluorophenoxy)phenyl)-2-(1...)
Affinity DataIC50:  248nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345667(CHEMBL1784808 | N-(3-(1H-imidazol-1-yl)propyl)-3-t...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345644(CHEMBL1784788 | E/Z-1-(2,4-dichlorophenyl)-3-pheny...)
Affinity DataIC50:  441nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345658(5-(8-methoxy-3,4-dihydro-2H-benzo[b][1,4]dioxepin-...)
Affinity DataIC50:  498nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345673(CHEMBL1784813 | N-(3-(1H-imidazol-1-yl)propyl)-2,2...)
Affinity DataIC50:  499nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345663(CHEMBL1784806 | N-(3-(1H-imidazol-1-yl)propyl)-4-e...)
Affinity DataIC50:  761nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345650(CHEMBL1784793 | rac-N-(1-(2,3-dihydrobenzo[b][1,4]...)
Affinity DataIC50:  991nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345661(CHEMBL1521315 | N-(3-(1H-imidazol-1-yl)propyl)-4-m...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345668(CHEMBL1538978 | N-(3-(1H-imidazol-1-yl)propyl)-4-(...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345656(CHEMBL1784800 | rac-2-((1H-1,2,4-triazol-1-yl)meth...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345654(CHEMBL1784797 | trans-3-(1H-imidazol-1-yl)-N-((4-(...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345653(CHEMBL1784796 | rac-1-(1H-imidazol-1-yl)-3-(4-((2-...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345649(1'-(2-(1H-1,2,4-triazol-1-yl)acetyl)-7-methoxyspir...)
Affinity DataIC50:  5.79E+3nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345662(CHEMBL1389987 | N-(3-(1H-imidazol-1-yl)propyl)-6-m...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345651(CHEMBL1784794 | rac-N-(2-(1H-1,2,4-triazol-1-yl)pr...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345670(CHEMBL1784810 | N-(2-(4-fluorophenoxy)phenyl)-2-me...)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345647(CHEMBL1784790 | rac-7-(2-hydroxy-3-(1H-1,2,4-triaz...)
Affinity DataIC50:  2.17E+4nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universita` Di Modena E Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50345652(CHEMBL1784795 | rac-N-(2-(1H-1,2,4-triazol-1-yl)pr...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed