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Found 9 with Last Name = 'capurro' and Initial = 'v'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Angelini

Curated by ChEMBL
LigandPNGBDBM186204(US9163013, 21)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Angelini

Curated by ChEMBL
LigandPNGBDBM186202(US9163013, 19)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Angelini

Curated by ChEMBL
LigandPNGBDBM186200(US9163013, 17)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Angelini

Curated by ChEMBL
LigandPNGBDBM50134914(CHEMBL3735730)
Affinity DataIC50:  210nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 7(Homo sapiens (Human))
Angelini

Curated by ChEMBL
LigandPNGBDBM50134187(CHEMBL3735506 | US11472795, Example C | US9611249,...)
Affinity DataIC50:  220nMAssay Description:Inhibition of human recombinant ERK5 by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Angelini

Curated by ChEMBL
LigandPNGBDBM186201(US9163013, 18)
Affinity DataIC50:  300nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Angelini

Curated by ChEMBL
LigandPNGBDBM50134187(CHEMBL3735506 | US11472795, Example C | US9611249,...)
Affinity DataIC50:  530nMAssay Description:Inhibition of human recombinant DYRK2 by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Angelini

Curated by ChEMBL
LigandPNGBDBM50134188(CHEMBL3735095)
Affinity DataIC50:  530nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Angelini

Curated by ChEMBL
LigandPNGBDBM50134187(CHEMBL3735506 | US11472795, Example C | US9611249,...)
Affinity DataIC50:  530nMAssay Description:Inhibition of human recombinant GRK2 by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed