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Found 52 with Last Name = 'carr' and Initial = 'aa'
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50000483((BRL 43694)1-Methyl-1H-indazole-3-carboxylic acid ...)
Affinity DataKi:  0.589nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  0.603nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor entirely in guinea pig ileumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKi:  1nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptors in the rabbit heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKi:  1.40nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  3.31nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptors in the rabbit heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50000483((BRL 43694)1-Methyl-1H-indazole-3-carboxylic acid ...)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM82561(CAS_40796-97-2 | TROPANYL 3,5-DICHLOROBENZOATE | T...)
Affinity DataKi:  55nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptors in the rabbit heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  87nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  88nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  128nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM48320(4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-metho...)
Affinity DataKi:  200nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor entirely in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM48320(4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-metho...)
Affinity DataKi:  229nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  540nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  2.25E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  5.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  6.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50283435((4,5-Dihydro-1H-imidazol-2-yl)-(3,3-diphenyl-propy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283436((4,5-Dihydro-1H-imidazol-2-yl)-(2,2-diphenyl-ethyl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283434((2,5-Dihydro-1H-benzo[e][1,3]diazepin-3-yl)-(3,3-d...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283433((2,2-Diphenyl-ethyl)-(1-methyl-4,5-dihydro-1H-imid...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283432(Benzhydryl-(4,5-dihydro-1H-imidazol-2-yl)-amine | ...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283431((2,2-Diphenyl-ethyl)-(3aS,7aS)-3a,4,5,6,7,7a-hexah...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283430((3,3-Diphenyl-propyl)-(3aS,7aS)-3a,4,5,6,7,7a-hexa...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283429((3,3-Diphenyl-propyl)-(1-methyl-4,5-dihydro-1H-imi...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283428((3,3-Diphenyl-propyl)-(4,5,6,7-tetrahydro-1H-[1,3]...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283427((2,2-Diphenyl-ethyl)-(1,4,5,6-tetrahydro-pyrimidin...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283426((4,4-Diphenyl-butyl)-(1-methyl-4,5-dihydro-1H-imid...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283425((2,2-Diphenyl-ethyl)-((E)-1,4,5,6,7,8-hexahydro-[1...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50004704((+)-cis-Diltiazem | (2S,3S)-5-(2-(dimethylamino)et...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283421(((E)-Azacyclotridec-1-en-2-yl)-(2,2-diphenyl-penty...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283417((3,3-Diphenyl-propyl)-(1-methyl-1,4,5,6-tetrahydro...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283418((3,3-Diphenyl-propyl)-((E)-1,4,5,6,7,8-hexahydro-[...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283419((2,5-Dihydro-1H-benzo[e][1,3]diazepin-3-yl)-(2,2-d...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283422((3,3-Diphenyl-propyl)-(1,4,5,6-tetrahydro-pyrimidi...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283423((2,2-Diphenyl-ethyl)-(1-methyl-1,4,5,6-tetrahydro-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283424((2,2-Diphenyl-ethyl)-(4,5,6,7-tetrahydro-1H-[1,3]d...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283420(((E)-Azacyclotridec-1-en-2-yl)-((1S,2S)-2-phenyl-c...)
Affinity DataEC50:  61nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283420(((E)-Azacyclotridec-1-en-2-yl)-((1S,2S)-2-phenyl-c...)
Affinity DataEC50:  61nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283421(((E)-Azacyclotridec-1-en-2-yl)-(2,2-diphenyl-penty...)
Affinity DataEC50:  61nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 3A/3B(Mus musculus (house mouse))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50000483((BRL 43694)1-Methyl-1H-indazole-3-carboxylic acid ...)
Affinity DataKd:  1.40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor was determined by using [3H]-ICS 205-930 as radioligand in mouse N1E 115 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Mus musculus (house mouse))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM48320(4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-metho...)
Affinity DataKd:  224nMAssay Description:Potency to 5-hydroxytryptamine 3 receptor entirely in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50283421(((E)-Azacyclotridec-1-en-2-yl)-(2,2-diphenyl-penty...)
Affinity DataEC50:  34nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 3A/3B(Mus musculus (house mouse))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKd:  2nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptors in the rabbit heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Mus musculus (house mouse))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50449568(CHEMBL2448558)
Affinity DataKd:  3.20nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Mus musculus (house mouse))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50227350(NORTROPISETRON | SDZ-206-792)
Affinity DataKd:  0.724nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Mus musculus (house mouse))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKd:  13nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Mus musculus (house mouse))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKd:  0.813nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
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