Affinity DataKi: 90nMAssay Description:Inhibition of factor 7a (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Inhibition of factor 7a (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:Inhibition of factor 7a (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of thrombin (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 452nMAssay Description:Inhibition of thrombin (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Inhibition of thrombin (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.32E+3nMAssay Description:Inhibition of factor 7a (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: >5.10E+3nMAssay Description:Inhibition of thrombin (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of glucocorticoid receptor-glucocorticoid complex transfected in rat R1 cells assessed as down-regulation of TPA-responsive element proinf...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Displacement of [3H]naloxone from kappa opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Griffith University
Curated by ChEMBL
Griffith University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of Pim2 kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Griffith University
Curated by ChEMBL
Griffith University
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of GST-tagged MAPKAPK2 assessed as [33P] incorporation after 40 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of Helicobacter pylori His-tagged ASD assessed as inhibition of phosphorylation of aspartate semialdehydeMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of carboxypeptidase BMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Binding affinity to glucocorticoid receptor by GR binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of factor 11a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.55E+3nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+3nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Griffith University
Curated by ChEMBL
Griffith University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
TargetProtein-S-isoprenylcysteine O-methyltransferase(Homo sapiens (Human))
Griffith University
Curated by ChEMBL
Griffith University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of [3H]SAM from Icmt relative to SAHMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.74E+3nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Griffith University
Curated by ChEMBL
Griffith University
Curated by ChEMBL
Affinity DataIC50: 3.71E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90E+3nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+4nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Binding affinity to glucocorticoid receptor by GR binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+4nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membranesMore data for this Ligand-Target Pair
TargetProtein-S-isoprenylcysteine O-methyltransferase(Homo sapiens (Human))
Griffith University
Curated by ChEMBL
Griffith University
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Icmt using [3H]SAM as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.46E+4nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsMore data for this Ligand-Target Pair