TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of human recombinant MAOB by amplex red assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of human recombinant MAO-B after 15 minsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 99nMAssay Description:Inhibition of human recombinant MAOB using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 195nMAssay Description:Inhibition of human recombinant MAOB by amplex red assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 195nMAssay Description:Inhibition of human recombinant MAO-B after 15 minsMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Rattus norvegicus)
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of rat BCATcMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 225nMAssay Description:Inhibition of human recombinant MAO-B after 15 minsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 228nMAssay Description:Inhibition of human recombinant MAOB using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 242nMAssay Description:Inhibition of human recombinant MAOB using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 268nMAssay Description:Inhibition of human recombinant MAOA using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 298nMAssay Description:Inhibition of human recombinant MAO-B after 15 minsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 305nMAssay Description:Inhibition of human recombinant MAOB using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of human recombinant MAOA assessed as inhibition of kynuramine conversion to fluorescent metabolite 4-hydroxyquinoline by fluorimetryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 709nMAssay Description:Inhibition of human recombinant MAOA using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant MAOB by amplex red assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 832nMAssay Description:Inhibition of human recombinant MAO-B after 15 minsMore data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Displacement of [3H]-rosiglitazone from human recombinant C-terminal His-tagged cytosolic domain of mitoNEET (32-108) by scintillation proximity assa...More data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Rattus norvegicus)
Northeastern Ohio Universities
Curated by ChEMBL
Northeastern Ohio Universities
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Displacement of [3H]rosiglitazone from rat liver mitochondrial mitoNEET by scintillation countingMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 921nMAssay Description:Inhibition of human recombinant MAOB using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 979nMAssay Description:Inhibition of human recombinant MAOA using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Rattus norvegicus)
Northeastern Ohio Universities
Curated by ChEMBL
Northeastern Ohio Universities
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]rosiglitazone from rat liver mitochondrial mitoNEET by scintillation countingMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of human recombinant MAOB by amplex red assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human recombinant MAOA assessed as inhibition of kynuramine conversion to fluorescent metabolite 4-hydroxyquinoline by fluorimetryMore data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Rattus norvegicus)
Northeastern Ohio Universities
Curated by ChEMBL
Northeastern Ohio Universities
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]rosiglitazone from rat liver mitochondrial mitoNEET by scintillation countingMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 1.73E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human recombinant C-terminal His-tagged cytosolic domain of mitoNEET (32-108) by scintillation proximity assa...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of human recombinant MAO-B after 15 minsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.29E+3nMAssay Description:Inhibition of human recombinant MAO-B after 15 minsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.29E+3nMAssay Description:Inhibition of human recombinant MAOB by amplex red assayMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of human recombinant MAOB by amplex red assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.49E+3nMAssay Description:Inhibition of human recombinant MAOB by amplex red assayMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.62E+3nMAssay Description:Inhibition of human recombinant MAOB using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 2.93E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human recombinant C-terminal His-tagged cytosolic domain of mitoNEET (32-108) by scintillation proximity assa...More data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, mitochondrial(Rattus norvegicus)
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rat BCATmMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 3.26E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human recombinant C-terminal His-tagged cytosolic domain of mitoNEET (32-108) by scintillation proximity assa...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy
Curated by ChEMBL
Affinity DataIC50: 3.35E+3nMAssay Description:Inhibition of human recombinant MAOB using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 3.36E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human recombinant C-terminal His-tagged cytosolic domain of mitoNEET (32-108) by scintillation proximity assa...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 3.49E+3nMAssay Description:Inhibition of human recombinant MAOA assessed as inhibition of kynuramine conversion to fluorescent metabolite 4-hydroxyquinoline by fluorimetryMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 4.47E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human recombinant C-terminal His-tagged cytosolic domain of mitoNEET (32-108) by scintillation proximity assa...More data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 4.98E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human recombinant C-terminal His-tagged cytosolic domain of mitoNEET (32-108) by scintillation proximity assa...More data for this Ligand-Target Pair
TargetCDGSH iron-sulfur domain-containing protein 1(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 5.23E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human recombinant C-terminal His-tagged cytosolic domain of mitoNEET (32-108) by scintillation proximity assa...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Northeast Ohio Medical University
Curated by ChEMBL
Northeast Ohio Medical University
Curated by ChEMBL
Affinity DataIC50: 5.36E+3nMAssay Description:Inhibition of human recombinant MAOA using kynuramine as substrate by fluorimetryMore data for this Ligand-Target Pair
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair