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Found 200 with Last Name = 'carson' and Initial = 'da'
TargetAdenosine kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  30nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50368712(CHEMBL608051)
Affinity DataKi:  40nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50368710(CHEMBL607761)
Affinity DataKi:  150nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50368709(CHEMBL607766)
Affinity DataKi:  160nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50368707(CHEMBL612205)
Affinity DataKi:  170nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50368708(CHEMBL611890)
Affinity DataKi:  300nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50368706(CHEMBL607762)
Affinity DataKi:  8.50E+3nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081323(4-(4-Bromo-6,7-dihydroxy-1-oxo-1H-isoquinolin-2-yl...)
Affinity DataIC50:  1.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081305(4-(6,7-Dihydroxy-1-oxo-1H-isoquinolin-2-yl)-butyri...)
Affinity DataIC50:  2.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081327(4-(6,7-Dimethoxy-4-oxo-4H-quinazolin-3-yl)-butyric...)
Affinity DataIC50:  3.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048928(4-(2,4-Dioxo-1-propyl-1,4-dihydro-2H-pteridin-3-yl...)
Affinity DataIC50:  3.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081304(4-(6-Amino-4-oxo-4H-quinazolin-3-yl)-butyric acid ...)
Affinity DataIC50:  4.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048929(4-(7-Methyl-2,6-dioxo-3-propyl-2,3,6,7-tetrahydro-...)
Affinity DataIC50:  5.00E+3nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048928(4-(2,4-Dioxo-1-propyl-1,4-dihydro-2H-pteridin-3-yl...)
Affinity DataIC50:  5.00E+3nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081354(4-(7-Amino-4-oxo-1,4-dihydro-2H-quinazolin-3-yl)-b...)
Affinity DataIC50:  5.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081335(4-(6,7-Dimethoxy-1-oxo-1H-isoquinolin-2-yl)-butyri...)
Affinity DataIC50:  5.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081326(4-(1-Oxo-1H-isoquinolin-2-yl)-butyric acid ethyl e...)
Affinity DataIC50:  5.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081306(4-(4-Cyano-6,7-dimethoxy-1-oxo-1H-isoquinolin-2-yl...)
Affinity DataIC50:  5.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048933(4-(3,7-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-purin...)
Affinity DataIC50:  6.00E+3nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081303(5-(6,7-Dimethoxy-4-oxo-4H-quinazolin-3-yl)-pentano...)
Affinity DataIC50:  6.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081333(4-(6,7-Diacetoxy-1-oxo-1H-isoquinolin-2-yl)-butyri...)
Affinity DataIC50:  9.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081343(4-(7-Amino-4-oxo-4H-quinazolin-3-yl)-butyric acid ...)
Affinity DataIC50:  9.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081351(3-(6,7-Dimethoxy-4-oxo-4H-quinazolin-3-yl)-propion...)
Affinity DataIC50:  9.00E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048931(3-(3,7-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-purin...)
Affinity DataIC50:  1.00E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081310(4-(6,7-Dimethoxy-1-oxo-1H-isoquinolin-2-yl)-butyri...)
Affinity DataIC50:  1.00E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081314(4-(6-Amino-4-oxo-1,4-dihydro-2H-quinazolin-3-yl)-b...)
Affinity DataIC50:  1.00E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048924(5-(3,7-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-purin...)
Affinity DataIC50:  1.10E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081330(4-(6,7-Bis-ethoxycarbonyloxy-1-oxo-1H-isoquinolin-...)
Affinity DataIC50:  1.10E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081352(4-(6,7-Dimethoxy-5-nitro-4-oxo-4H-quinazolin-3-yl)...)
Affinity DataIC50:  1.10E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  1.20E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048943(4-(1-Methyl-2,4-dioxo-1,4-dihydro-2H-pteridin-3-yl...)
Affinity DataIC50:  1.20E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081353(4-(4-Aminomethyl-6,7-dimethoxy-1-oxo-1H-isoquinoli...)
Affinity DataIC50:  1.30E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081355(4-(2-Azido-6,7-dimethoxy-4-oxo-4H-quinazolin-3-yl)...)
Affinity DataIC50:  1.40E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048925(4-(1-Butyl-2,4-dioxo-1,4-dihydro-2H-pteridin-3-yl)...)
Affinity DataIC50:  1.50E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081322(4-(4-Acetyl-6,7-dimethoxy-1-oxo-1H-isoquinolin-2-y...)
Affinity DataIC50:  1.50E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081312(4-(5-Amino-6,7-dimethoxy-4-oxo-4H-quinazolin-3-yl)...)
Affinity DataIC50:  1.50E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048932(4-(2,4-Dioxo-1-pentyl-1,4-dihydro-2H-pteridin-3-yl...)
Affinity DataIC50:  1.60E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048935(4-(5,7-Dioxo-4-propyl-4,5-dihydro-7H-[1,2,5]thiadi...)
Affinity DataIC50:  1.80E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048920(4-[2,4-Dioxo-1-(tetrahydro-furan-3-yl)-1,4-dihydro...)
Affinity DataIC50:  1.90E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081312(4-(5-Amino-6,7-dimethoxy-4-oxo-4H-quinazolin-3-yl)...)
Affinity DataIC50:  2.00E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081328(4-(4-Fluoro-6,7-dimethoxy-1-oxo-1H-isoquinolin-2-y...)
Affinity DataIC50:  2.00E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048948(4-(1-Isobutyl-2,4-dioxo-1,4-dihydro-2H-pteridin-3-...)
Affinity DataIC50:  2.00E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081342(5-(6,7-Dimethoxy-1-oxo-1H-isoquinolin-2-yl)-pentan...)
Affinity DataIC50:  2.10E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081319(4-(5-Chloro-6,7-dimethoxy-4-oxo-4H-quinazolin-3-yl...)
Affinity DataIC50:  2.20E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048938((Z)-4-(1-Methyl-2,4-dioxo-1,4-dihydro-2H-pteridin-...)
Affinity DataIC50:  2.50E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50048942(4-(4-Methyl-5,7-dioxo-4,5-dihydro-7H-[1,2,5]thiadi...)
Affinity DataIC50:  2.50E+4nMAssay Description:TNF-alpha production in PBMC by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081307(4-(2-Dimethylamino-6,7-dimethoxy-quinazolin-4-ylox...)
Affinity DataIC50: >2.50E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081308(4-(6,7-Dimethoxy-4-oxo-2-phenylamino-4H-quinazolin...)
Affinity DataIC50: >2.50E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081309(4-(6-Nitro-4-oxo-4H-quinazolin-3-yl)-butyric acid ...)
Affinity DataIC50: >2.50E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50081316(4-(7-Fluoro-4-oxo-4H-quinazolin-3-yl)-butyric acid...)
Affinity DataIC50: >2.50E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against Tumor necrosis factor alpha from human PMBC cell line by ELISA test.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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