TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataIC50: 6.74E+3nMAssay Description:Inhibition of human CKalpha1 assessed as reduction in 14C incorporation from [methyl-14C]choline to phosphatidylcholine using [methyl-14C]choline as ...More data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human CKalpha1 assessed as reduction in 14C incorporation from [methyl-14C]choline to phosphatidylcholine using [methyl-14C]choline as ...More data for this Ligand-Target Pair
Affinity DataEC50: 6.71E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.58E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+4nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.61E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.07E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.51E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.75E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.27E+4nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.20E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.96E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.31E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.96E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.09E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.45E+4nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.93E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.79E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.02E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 1.40E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 2.40E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 890nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 670nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 370nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 185nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 3.50E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 4.90E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 4.50E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 8.20E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 3.30E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 3.60E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 6.30E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Affinity DataEC50: 1.64E+4nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.11E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair