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Found 40 with Last Name = 'castro navas' and Initial = 'ff'
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556491(CHEMBL4784458)
Affinity DataIC50:  6.74E+3nMAssay Description:Inhibition of human CKalpha1 assessed as reduction in 14C incorporation from [methyl-14C]choline to phosphatidylcholine using [methyl-14C]choline as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556492(CHEMBL4747352)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of human CKalpha1 assessed as reduction in 14C incorporation from [methyl-14C]choline to phosphatidylcholine using [methyl-14C]choline as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM20177((1S,2R,5S,10S,11S,14R,15S)-14-[(2S,3R)-3-hydroxy-6...)
Affinity DataEC50:  6.71E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257931(CHEMBL4073435)
Affinity DataEC50:  5.58E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257932(CHEMBL4085972)
Affinity DataEC50:  1.58E+4nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257933(CHEMBL4086897)
Affinity DataEC50:  6.61E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257934(CHEMBL4104778)
Affinity DataEC50:  8.07E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257935(CHEMBL4067156)
Affinity DataEC50:  3.20E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257936(CHEMBL4059545)
Affinity DataEC50:  8.51E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM20177((1S,2R,5S,10S,11S,14R,15S)-14-[(2S,3R)-3-hydroxy-6...)
Affinity DataEC50:  4.75E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257930(CHEMBL4061349)
Affinity DataEC50:  1.27E+4nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257929(CHEMBL4097209)
Affinity DataEC50:  7.20E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257928(CHEMBL4070016)
Affinity DataEC50:  1.96E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257937(CHEMBL4094610)
Affinity DataEC50:  2.31E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257933(CHEMBL4086897)
Affinity DataEC50:  1.96E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257938(CHEMBL4089508)
Affinity DataEC50:  2.09E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257939(CHEMBL4078083)
Affinity DataEC50:  1.45E+4nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257937(CHEMBL4094610)
Affinity DataEC50:  6.93E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257938(CHEMBL4089508)
Affinity DataEC50:  3.79E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257935(CHEMBL4067156)
Affinity DataEC50:  2.70E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257939(CHEMBL4078083)
Affinity DataEC50:  6.02E+3nMAssay Description:Activation of GAL4 fused human LXR beta expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556486(CHEMBL1508421)
Affinity DataKd:  1.40E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50342854(1-Benzyl-4-(pyrrolidin-1-yl)pyridinium Bromide | C...)
Affinity DataKd:  2.40E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556487(CHEMBL4763249)
Affinity DataKd:  400nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556488(CHEMBL4756022)
Affinity DataKd:  890nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556489(CHEMBL4755703)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556490(CHEMBL4748826)
Affinity DataKd:  670nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556491(CHEMBL4784458)
Affinity DataKd:  370nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556492(CHEMBL4747352)
Affinity DataKd:  185nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556493(CHEMBL3561645)
Affinity DataKd:  3.50E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556494(CHEMBL4754833)
Affinity DataKd:  4.90E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556495(CHEMBL4796843)
Affinity DataKd:  4.50E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556496(CHEMBL4776753)
Affinity DataKd:  8.20E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556487(CHEMBL4763249)
Affinity DataKd:  3.30E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556488(CHEMBL4756022)
Affinity DataKd:  3.60E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556491(CHEMBL4784458)
Affinity DataKd:  6.30E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556492(CHEMBL4747352)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257930(CHEMBL4061349)
Affinity DataEC50:  1.64E+4nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257928(CHEMBL4070016)
Affinity DataEC50:  1.50E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257929(CHEMBL4097209)
Affinity DataEC50:  4.11E+3nMAssay Description:Activation of GAL4 fused human LXR alpha expressed in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed