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Found 63 with Last Name = 'cepa' and Initial = 'sp'
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371080(CHEMBL376392)
Affinity DataIC50:  1nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371071(CHEMBL227205)
Affinity DataIC50:  3nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371087(CHEMBL375514)
Affinity DataIC50:  4nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371060(CHEMBL226646)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371053(CHEMBL227256)
Affinity DataIC50:  5nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371046(CHEMBL427416)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371059(CHEMBL227313)
Affinity DataIC50:  6nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371077(CHEMBL227255)
Affinity DataIC50:  7nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371084(CHEMBL227257)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371074(CHEMBL388735)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371043(CHEMBL375265)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371073(CHEMBL226648)
Affinity DataIC50:  9.20nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371051(CHEMBL227280)
Affinity DataIC50:  10nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371050(CHEMBL376117)
Affinity DataIC50:  10nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371048(CHEMBL227281)
Affinity DataIC50:  10nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371058(CHEMBL227269)
Affinity DataIC50:  10nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371079(CHEMBL442055)
Affinity DataIC50:  10nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371069(CHEMBL226597)
Affinity DataIC50:  12nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371088(CHEMBL229271)
Affinity DataIC50:  12nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371047(CHEMBL229328)
Affinity DataIC50:  14nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371064(CHEMBL227204)
Affinity DataIC50:  16nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371056(CHEMBL229327)
Affinity DataIC50:  19nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371081(CHEMBL226702)
Affinity DataIC50:  20nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371044(CHEMBL390518)
Affinity DataIC50:  20nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371054(CHEMBL229270)
Affinity DataIC50:  20nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371067(CHEMBL375954)
Affinity DataIC50:  21nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371065(CHEMBL227217)
Affinity DataIC50:  24nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371070(CHEMBL227282)
Affinity DataIC50:  26nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371085(CHEMBL226701)
Affinity DataIC50:  32nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371062(CHEMBL227203)
Affinity DataIC50:  34nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50506590(CHEMBL4593992)
Affinity DataIC50:  41nMAssay Description:Inhibition of C-terminal 8-His tagged wild type human IDH1 (1 to 414 residues) expressed in Escherichia coli BL21(DE3)-T1R preincubated for 15 mins u...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371063(CHEMBL227258)
Affinity DataIC50:  57nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371040(CHEMBL226691)
Affinity DataIC50:  60nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371075(CHEMBL390818)
Affinity DataIC50:  63nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371041(CHEMBL229326)
Affinity DataIC50:  65nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371078(CHEMBL227270)
Affinity DataIC50:  70nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50506594(CHEMBL4556998)
Affinity DataIC50:  82nMAssay Description:Inhibition of C-terminal 8-His tagged wild type human IDH1 (1 to 414 residues) expressed in Escherichia coli BL21(DE3)-T1R preincubated for 15 mins u...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371083(CHEMBL388413)
Affinity DataIC50:  85nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50506592(CHEMBL4535154)
Affinity DataIC50:  110nMAssay Description:Inhibition of C-terminal 8-His tagged wild type human IDH1 (1 to 414 residues) expressed in Escherichia coli BL21(DE3)-T1R preincubated for 15 mins u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50506585(CHEMBL4515358)
Affinity DataIC50:  120nMAssay Description:Inhibition of C-terminal 8-His tagged wild type human IDH1 (1 to 414 residues) expressed in Escherichia coli BL21(DE3)-T1R preincubated for 15 mins u...More data for this Ligand-Target Pair
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371086(CHEMBL227152)
Affinity DataIC50:  150nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50506593(CHEMBL4540440)
Affinity DataIC50:  210nMAssay Description:Inhibition of C-terminal 8-His tagged wild type human IDH1 (1 to 414 residues) expressed in Escherichia coli BL21(DE3)-T1R preincubated for 15 mins u...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371089(CHEMBL226692)
Affinity DataIC50:  220nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371049(CHEMBL227206)
Affinity DataIC50:  250nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50506584(CHEMBL221360)
Affinity DataIC50:  270nMAssay Description:Inhibition of C-terminal 8-His tagged wild type human IDH1 (1 to 414 residues) expressed in Escherichia coli BL21(DE3)-T1R preincubated for 15 mins u...More data for this Ligand-Target Pair
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371055(CHEMBL226647)
Affinity DataIC50:  370nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371068(CHEMBL229269)
Affinity DataIC50:  394nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50506591(CHEMBL4548727)
Affinity DataIC50:  410nMAssay Description:Inhibition of C-terminal 8-His tagged wild type human IDH1 (1 to 414 residues) expressed in Escherichia coli BL21(DE3)-T1R preincubated for 15 mins u...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371052(CHEMBL229254)
Affinity DataIC50:  505nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50371042(CHEMBL229212)
Affinity DataIC50:  627nMAssay Description:Inhibition of SCD1 in ob/ob mouse liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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