Affinity DataIC50: 3nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 96nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataIC50: 106nMAssay Description:Displacement of [3H]E2 from ERbeta ligand binding domainMore data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 112nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 117nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 164nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
Affinity DataIC50: 165nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
Affinity DataIC50: 196nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 198nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 206nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop
Curated by ChEMBL
Sanofi Winthrop
Curated by ChEMBL
Affinity DataIC50: 213nMAssay Description:Inhibition of outward potassium currents (IKn) in human T-lymphocyte N-type potassium channels.More data for this Ligand-Target Pair