Compile Data Set for Download or QSAR
maximum 50k data
Found 174 with Last Name = 'chadwick' and Initial = 'cc'
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157485(4-[1-isopropyl-7-(trifluoromethyl)-1H-indazol-3-yl...)
Affinity DataIC50:  3nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177756(CHEMBL202472 | N-(2,6-diethylphenyl)-4-hydroxy-3-m...)
Affinity DataIC50:  5nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177740(CHEMBL371637 | N-(2-ethyl-6-methylphenyl)-4-hydrox...)
Affinity DataIC50:  7nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177763(CHEMBL201834 | N-(2,6-dimethylphenyl)-4-hydroxy-3-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157496(4-[1-(2,5-dichlorophenyl)-6-hydroxy-1H-indazol-3-y...)
Affinity DataIC50:  15nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177752(CHEMBL202607 | N-(2,6-dichlorophenyl)-4-hydroxy-3-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157483(4-(1-cyclopentyl-7-fluoro-1H-indazol-3-yl)phenol |...)
Affinity DataIC50:  18nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157488(4-(7-chloro-1-cyclopentyl-1H-indazol-3-yl)phenol |...)
Affinity DataIC50:  18nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157501(4-[1-isopropyl-7-(trifluoromethyl)-1H-indazol-3-yl...)
Affinity DataIC50:  20nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177764(CHEMBL383691 | N-(2-chloro-6-methylphenyl)-4-hydro...)
Affinity DataIC50:  24nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157498(4-(1-butyl-7-chloro-1H-indazol-3-yl)phenol | CHEMB...)
Affinity DataIC50:  25nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177748(CHEMBL202500 | N-(2-chloro-6-methylphenyl)-4-hydro...)
Affinity DataIC50:  26nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177746(CHEMBL202624 | N-(2-bromophenyl)-4-hydroxy-N-propy...)
Affinity DataIC50:  26nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157491(4-[1-(2,5-difluorophenyl)-6-hydroxy-1H-indazol-3-y...)
Affinity DataIC50:  31nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030498(CHEMBL53841 | [1-Benzyl-7-chloro-1H-quinolin-(4E)-...)
Affinity DataIC50:  32nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157504(4-(7-chloro-1-cyclohexyl-1H-indazol-3-yl)phenol | ...)
Affinity DataIC50:  37nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157489(4-[1-(3-fluorophenyl)-6-hydroxy-1H-indazol-3-yl]be...)
Affinity DataIC50:  39nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157503(4-(7-methyl-1-propyl-1H-indazol-3-yl)phenol | CHEM...)
Affinity DataIC50:  40nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157500(4-[6-hydroxy-1-(4-methylphenyl)-1H-indazol-3-yl]be...)
Affinity DataIC50:  40nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177749(CHEMBL202155 | N-(2-bromophenyl)-4-hydroxy-3-methy...)
Affinity DataIC50:  40nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177757(CHEMBL264655 | N-(2-chlorophenyl)-4-hydroxy-N-prop...)
Affinity DataIC50:  42nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030511(CHEMBL293721 | [1-Benzyl-6-methoxy-1H-quinolin-(4E...)
Affinity DataIC50:  47nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157486(4-(6-HYDROXY-1H-INDAZOL-3-YL)BENZENE-1,3-DIOL | CH...)
Affinity DataIC50:  48nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157508(4-[1-(3-chlorophenyl)-6-hydroxy-1H-indazol-3-yl]be...)
Affinity DataIC50:  50nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177744(CHEMBL204185 | N-(2-chlorophenyl)-4-hydroxy-3-meth...)
Affinity DataIC50:  51nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157502(4-(7-chloro-1-propyl-1H-indazol-3-yl)phenol | CHEM...)
Affinity DataIC50:  52nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177736(4-hydroxy-N-propyl-N-(2-(trifluoromethyl)phenyl)be...)
Affinity DataIC50:  54nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157507(4-[1-allyl-7-(trifluoromethyl)-1H-indazol-3-yl]-3-...)
Affinity DataIC50:  59nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177760(CHEMBL372997 | N-(2-bromophenyl)-4-hydroxy-N-propy...)
Affinity DataIC50:  60nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157487(4-(6-hydroxy-1-propyl-1H-indazol-3-yl)benzene-1,3-...)
Affinity DataIC50:  62nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030510(CHEMBL299668 | [1-Benzyl-7-chloro-1H-quinolin-(4E)...)
Affinity DataIC50:  65nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177755(CHEMBL203565 | N-(2-fluorophenyl)-4-hydroxy-N-prop...)
Affinity DataIC50:  74nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030505(CHEMBL56589 | [7-Chloro-1-naphthalen-2-yl-1H-quino...)
Affinity DataIC50:  75nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030495(CHEMBL55202 | [7-Chloro-1-(4-methoxy-benzyl)-1H-qu...)
Affinity DataIC50:  88nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177762(CHEMBL202248 | N-(2-bromophenyl)-N-ethyl-4-hydroxy...)
Affinity DataIC50:  90nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157493(4-[1-allyl-7-(trifluoromethyl)-1H-indazol-3-yl]ben...)
Affinity DataIC50:  93nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157505(4-[1-(2-hydroxyethyl)-7-(trifluoromethyl)-1H-indaz...)
Affinity DataIC50:  96nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030499(CHEMBL56998 | [7-Chloro-1-(4-chloro-benzyl)-1H-qui...)
Affinity DataIC50:  100nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157484(4-(1-benzyl-7-chloro-1H-indazol-3-yl)phenol | CHEM...)
Affinity DataIC50:  105nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157493(4-[1-allyl-7-(trifluoromethyl)-1H-indazol-3-yl]ben...)
Affinity DataIC50:  106nMAssay Description:Displacement of [3H]E2 from ERbeta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177753(4-hydroxy-3-methyl-N-propyl-N-o-tolylbenzenesulfon...)
Affinity DataIC50:  109nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157494(4-(1-butyl-6-hydroxy-1H-indazol-3-yl)benzene-1,3-d...)
Affinity DataIC50:  112nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030508(CHEMBL54934 | [1-Benzyl-7-chloro-1H-quinolin-(4E)-...)
Affinity DataIC50:  117nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030521(CHEMBL56173 | [1-Benzyl-1H-quinolin-(4E)-ylidene]-...)
Affinity DataIC50:  164nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157497(4-[6-hydroxy-1-(2,2,2-trifluoroethyl)-1H-indazol-3...)
Affinity DataIC50:  165nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030497(CHEMBL298622 | [7-Chloro-1-(2-chloro-benzyl)-1H-qu...)
Affinity DataIC50:  190nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157506(4-[1-benzyl-7-(trifluoromethyl)-1H-indazol-3-yl]ph...)
Affinity DataIC50:  196nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030500(CHEMBL293083 | [1-Benzyl-7-chloro-1H-quinolin-(4E)...)
Affinity DataIC50:  198nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030528(CHEMBL291738 | [1-Benzyl-7-chloro-1H-quinolin-(4E)...)
Affinity DataIC50:  206nMAssay Description:Concentration inhibiting [125I]-ChTX (charybdotoxin) binding to N-type potassium channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Sanofi Winthrop

Curated by ChEMBL
LigandPNGBDBM50030496(CHEMBL416313 | [1-(4-Chloro-benzyl)-6-trifluoromet...)
Affinity DataIC50:  213nMAssay Description:Inhibition of outward potassium currents (IKn) in human T-lymphocyte N-type potassium channels.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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