Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5.30E+3nMAssay Description:Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+5nMAssay Description:Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Binding affinity to LTB4 receptor in human U937 cells by whole cell assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Antagonist activity at LTB4 receptor in fura-2 loaded human U937 cells assessed as inhibition of LTB4-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+4nMAssay Description:Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membraneMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 4.46E+4nMAssay Description:Inhibition of DNA topoisomerase 2 assessed as bacteriophage P4 DNA unknotting after 30 minsMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 8.18E+4nMAssay Description:Inhibition of DNA topoisomerase 2 assessed as bacteriophage P4 DNA unknotting after 30 minsMore data for this Ligand-Target Pair