Compile Data Set for Download or QSAR
maximum 50k data
Found 112 with Last Name = 'chang' and Initial = 'cd'
TargetGTP:AMP phosphotransferase AK3, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50027422(1N-{4-[9-(3,4-dihydroxy-5-hydroxymethyltetrahydro-...)
Affinity DataKi:  9.00E+5nMAssay Description:Competitive inhibition of adenylate kinase II in rat liver with respect to ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50027422(1N-{4-[9-(3,4-dihydroxy-5-hydroxymethyltetrahydro-...)
Affinity DataKi:  1.10E+6nMAssay Description:Competitive inhibition of adenylate kinase III in rat liver with respect to ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323659(CHEMBL1208890 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  1nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323660(CHEMBL1208891 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  2nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50551233(CHEMBL4790152)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac)-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac)-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant human C-terminal FLAG-His-tagged HDAC1 (1 to 482 residues) expressed in Sf21 cells using RHK-K(Ac)-AMC as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50551231(CHEMBL4798549)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac)-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant human HDAC3 using RHK-K(Ac)-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323662(CHEMBL1208954 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  13nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274366(2-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-N-(4-(2-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human p38-alpha kinase phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  17nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274368(2-(5-tert-butyl-2-methylfuran-3-yl)-N-(4-(6-(morph...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human p38alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323668(CHEMBL1208953 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  21nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274367(2-(5-tert-butyl-2-methylfuran-3-yl)-N-(4-(2-morpho...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323666(CHEMBL1209013 | N-(5-tert-butyl-3-cyano-2-methoxyp...)
Affinity DataIC50:  22nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374798(CHEMBL255410)
Affinity DataIC50:  23nMAssay Description:Inhibition of human p38-alpha kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323660(CHEMBL1208891 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  25nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323650(CHEMBL1209838 | N-(3-cyano-5-morpholinophenyl)-2-(...)
Affinity DataIC50:  28nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM15244(5-(2,6-dichlorophenyl)-2-(2,4-difluorophenyl)sulfa...)
Affinity DataIC50:  29nMAssay Description:Inhibition of human p38-alpha kinaseMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50551227(CHEMBL4782478)
Affinity DataIC50:  33nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac)-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323649(CHEMBL1209837 | N-(3-tert-butyl-5-cyanophenyl)-2-(...)
Affinity DataIC50:  33nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323662(CHEMBL1208954 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  38nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323654(CHEMBL1208829 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  38nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  39nMAssay Description:Inhibition of human p38-alpha kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  39nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323651(CHEMBL1209839 | N-(5-tert-butyl-3-cyano-2-methoxyp...)
Affinity DataIC50:  42nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human p38-alpha kinaseMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50551232(CHEMBL4790559)
Affinity DataIC50:  44nMAssay Description:Inhibition of HSP90a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50551231(CHEMBL4798549)
Affinity DataIC50:  44nMAssay Description:Inhibition of HSP90a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  44nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50551234(CHEMBL4789155)
Affinity DataIC50:  47nMAssay Description:Inhibition of HSP90a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323661(CHEMBL1208952 | N-(5-tert-butyl-3-cyano-2-methoxyp...)
Affinity DataIC50:  51nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274364(2-(3-tert-butyl-1-m-tolyl-1H-pyrazol-5-yl)-2-(hydr...)
Affinity DataIC50:  59nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323654(CHEMBL1208829 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  59nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274368(2-(5-tert-butyl-2-methylfuran-3-yl)-N-(4-(6-(morph...)
Affinity DataIC50:  59nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323664(CHEMBL1208956 | N-(5-tert-butyl-3-cyano-2-methoxyp...)
Affinity DataIC50:  60nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM20800(2-amino-6-halopurine analogue, 20 | 6-chloro-9-[(4...)
Affinity DataIC50:  66nMAssay Description:Inhibition of HSP90a (unknown origin)More data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50551227(CHEMBL4782478)
Affinity DataIC50:  66nMAssay Description:Inhibition of HSP90a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50551229(CHEMBL4740842)
Affinity DataIC50:  69nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac)-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323653(CHEMBL1208828 | N-(5-tert-butyl-3-chloro-2-methoxy...)
Affinity DataIC50:  70nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274366(2-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-N-(4-(2-...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human p38alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323655(5-tert-butyl-N-cyclopropyl-2-methoxy-3-(2-(4-(2-mo...)
Affinity DataIC50:  71nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323659(CHEMBL1208890 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  72nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323663(CHEMBL1208955 | N-(5-tert-butyl-3-cyano-2-methoxyp...)
Affinity DataIC50:  78nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323658(CHEMBL1208889 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  90nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  99nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using fluorescence substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274364(2-(3-tert-butyl-1-m-tolyl-1H-pyrazol-5-yl)-2-(hydr...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human p38alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50551235(CHEMBL4747757)
Affinity DataIC50:  104nMAssay Description:Inhibition of HSP90a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 112 total ) | Next | Last >>
Jump to: