Compile Data Set for Download or QSAR
maximum 50k data
Found 314 with Last Name = 'cuzzupe' and Initial = 'a'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  2nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313798(US10167292, Example 42)
Affinity DataIC50:  2nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  3nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  3nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313789(US10167292, Example 33)
Affinity DataIC50:  4nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313798(US10167292, Example 42)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313797(US10167292, Example 41)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  9nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313796(US10167292, Example 40)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313778(US10167292, Example 13)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313803(US10167292, Example 47)
Affinity DataIC50:  11nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  11nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataIC50:  12nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313771(US10167292, Example 5)
Affinity DataIC50:  12nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  12nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313777(US10167292, Example 12)
Affinity DataIC50:  12nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313778(US10167292, Example 13)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313803(US10167292, Example 47)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313795(US10167292, Example 39)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313795(US10167292, Example 39)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313797(US10167292, Example 41)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313792(US10167292, Example 36)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313792(US10167292, Example 36)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313777(US10167292, Example 12)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313795(US10167292, Example 39)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313794(US10167292, Example 38)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313793(US10167292, Example 37)
Affinity DataIC50:  15nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313778(US10167292, Example 13)
Affinity DataIC50:  15nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313788(US10167292, Example 32)
Affinity DataIC50:  16nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataIC50:  16nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  16nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285938(CHEMBL4174918)
Affinity DataIC50:  17nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313789(US10167292, Example 33)
Affinity DataIC50:  17nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313798(US10167292, Example 42)
Affinity DataIC50:  17nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313788(US10167292, Example 32)
Affinity DataIC50:  17nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313787(US10167292, Example 31)
Affinity DataIC50:  18nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313792(US10167292, Example 36)
Affinity DataIC50:  18nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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