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Found 83 with Last Name = 'danahay' and Initial = 'h'
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246998(CHEMBL505558 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  12nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246999(CHEMBL500474 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  19nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246997(CHEMBL505738 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  27nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246995(CHEMBL505048 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  28nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247004((3R,5S)-5-(((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-...)
Affinity DataKi:  29nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246992(CHEMBL498914 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246994(CHEMBL443101 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  41nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246996(CHEMBL506226 | {(R)-1-[(2S,4R)-2-[(S)-5-Amino-1-(b...)
Affinity DataKi:  45nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246991(CHEMBL509770 | benzyl (R)-1-((2S,3S)-2-(((S)-6-ami...)
Affinity DataKi:  49nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247002(((R)-1-{(2S,4R)-2-[(S)-5-Amino-1-(benzooxazole-2-c...)
Affinity DataKi:  60nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247000(CHEMBL446259 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  65nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247005((3R,5S)-5-(((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-...)
Affinity DataKi:  101nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247001(CHEMBL448873 | Phenyl-carbamic acid (3R,5S)-5-[(S)...)
Affinity DataKi:  130nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247003(CHEMBL501945 | {(R)-1-[(2S,4R)-2-[(S)-5-Amino-1-(b...)
Affinity DataKi:  176nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246990(CHEMBL454436 | benzyl (R)-1-((2S,3R)-2-(((S)-6-ami...)
Affinity DataKi:  267nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247006((3R,5S)-5-((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-o...)
Affinity DataKi:  510nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246993(CHEMBL507245 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  1.04E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246989(CHEMBL501802 | benzyl (R)-1-((S)-2-(((S)-6-amino-1...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247007(((R)-1-{(2S,4R)-2-[(S)-5-Amino-1-(benzooxazole-2-c...)
Affinity DataKi:  1.55E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246988(CHEMBL503925 | benzyl (S)-1-((S)-1-((S)-6-amino-1-...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246986(CHEMBL507205 | benzyl (S)-1-((S)-1-((S)-6-amino-1-...)
Affinity DataKi:  5.72E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246987(CHEMBL504394 | benzyl (S)-6-amino-1-((S)-1-((S)-6-...)
Affinity DataKi:  5.78E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246985(CHEMBL507704 | benzyl (S)-6-amino-1-((S)-1-((S)-6-...)
Affinity DataKi:  1.52E+4nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246983(CHEMBL509923 | benzyl (S)-1-((S)-6-amino-1-(benzo[...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246984(CHEMBL508055 | benzyl (S)-1-((S)-6-amino-1-(benzo[...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50363361(CHEMBL1945199)
Affinity DataIC50:  330nMAssay Description:Binding affinity to human ERG channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50363361(CHEMBL1945199)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of human ERG channel by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataEC50:  8.20E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential preincubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581833(CHEMBL1949980)
Affinity DataEC50:  390nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential preincubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581834(CHEMBL5080252)
Affinity DataEC50:  920nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataEC50:  8.48E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581833(CHEMBL1949980)
Affinity DataEC50:  1.25E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581834(CHEMBL5080252)
Affinity DataEC50:  78nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581835(CHEMBL5085731)
Affinity DataEC50:  3.78E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581836(CHEBI:73244 | METHYL ANTHRANILATE)
Affinity DataEC50:  3.00E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581837(CHEMBL5083598)
Affinity DataEC50:  362nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581838(CHEMBL5085939)
Affinity DataEC50:  240nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581839(CHEMBL5076850)
Affinity DataEC50:  329nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581840(CHEMBL5091133)
Affinity DataEC50:  462nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581841(CHEMBL5085858)
Affinity DataEC50:  5.31E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581842(CHEMBL5077730)
Affinity DataEC50:  5.83E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581843(CHEMBL5085049)
Affinity DataEC50:  1.86E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581844(CHEMBL5077005)
Affinity DataEC50:  3.00E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581845(CHEMBL5086285)
Affinity DataEC50:  250nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581846(CHEMBL5093146)
Affinity DataEC50:  40nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581847(CHEMBL5082261)
Affinity DataEC50:  70nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581848(CHEMBL5081202)
Affinity DataEC50:  23nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581849(CHEMBL5087757)
Affinity DataEC50:  9nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM297398(3-Amino-6-bromo-5-trifluoromethyl-pyridine-2-carbo...)
Affinity DataEC50:  15nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM297396(3-Amino-6-bromo-5-trifluoromethyl-pyridine-2-carbo...)
Affinity DataEC50:  30nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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