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Found 95 with Last Name = 'dandekar' and Initial = 't'
TargetGlycine receptor subunit alpha-1(RAT)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]strychnine from glycine receptor alpha 1 in rat brain synaptic membranesMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(RAT)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]strychnine from glycine receptor alpha 1 in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232888(CHEMBL4096857)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataKi:  189nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)
Affinity DataKi:  241nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)
Affinity DataIC50:  43nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)
Affinity DataIC50:  46nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)
Affinity DataIC50:  49nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)
Affinity DataIC50:  52nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataIC50:  56nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50:  58nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)
Affinity DataIC50:  59nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataIC50:  75nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)
Affinity DataIC50:  76nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)
Affinity DataIC50:  77nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)
Affinity DataIC50:  78nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)
Affinity DataIC50:  80nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)
Affinity DataIC50:  82nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50:  93nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)
Affinity DataIC50:  95nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)
Affinity DataIC50:  97nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)
Affinity DataIC50:  97nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)
Affinity DataIC50:  98nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataIC50:  105nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)
Affinity DataIC50:  109nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)
Affinity DataIC50:  115nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)
Affinity DataIC50:  116nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)
Affinity DataIC50:  150nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232891(CHEMBL4086212)
Affinity DataIC50:  166nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232891(CHEMBL4086212)
Affinity DataIC50:  170nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50:  182nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232888(CHEMBL4096857)
Affinity DataIC50:  201nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataIC50:  214nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)
Affinity DataIC50:  214nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232887(CHEMBL4096505)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232887(CHEMBL4096505)
Affinity DataIC50:  224nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)
Affinity DataIC50:  240nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232895(CHEMBL4087535)
Affinity DataIC50:  245nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232895(CHEMBL4087535)
Affinity DataIC50:  250nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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