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Found 57 with Last Name = 'davis' and Initial = 'tp'
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069559(Biphalin Analogue | CHEMBL2371057)
Affinity DataKi:  0.790nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069560(Biphalin Analogue | CHEMBL2371080)
Affinity DataKi:  0.910nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069562(2-Amino-N-((S)-1-{[((R)-1-{N'-[(R)-2-(2-{(S)-2-[2-...)
Affinity DataKi:  1.30nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069563(Biphalin Analogue | CHEMBL2371079)
Affinity DataKi:  1.70nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069558(2-Amino-N-((S)-1-{[(2-{N'-[2-(2-{(S)-2-[2-amino-3-...)
Affinity DataKi:  2.80nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069561(2-Amino-N-((S)-1-{[((S)-1-{N'-[(S)-2-(2-{(S)-2-[2-...)
Affinity DataKi:  3nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069558(2-Amino-N-((S)-1-{[(2-{N'-[2-(2-{(S)-2-[2-amino-3-...)
Affinity DataKi:  5.20nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069559(Biphalin Analogue | CHEMBL2371057)
Affinity DataKi:  6.40nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069563(Biphalin Analogue | CHEMBL2371079)
Affinity DataKi:  7.40nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069560(Biphalin Analogue | CHEMBL2371080)
Affinity DataKi:  7.80nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069561(2-Amino-N-((S)-1-{[((S)-1-{N'-[(S)-2-(2-{(S)-2-[2-...)
Affinity DataKi:  11nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069562(2-Amino-N-((S)-1-{[((R)-1-{N'-[(R)-2-(2-{(S)-2-[2-...)
Affinity DataKi:  110nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069559(Biphalin Analogue | CHEMBL2371057)
Affinity DataIC50:  1.70nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069563(Biphalin Analogue | CHEMBL2371079)
Affinity DataIC50:  2.20nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50369571(CHEMBL1790710)
Affinity DataIC50:  2.40nMAssay Description:Binding affinity towards Opioid receptor delta 1 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50369571(CHEMBL1790710)
Affinity DataIC50:  2.70nMAssay Description:Opioid receptor activity was evaluated using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50369572(CHEMBL1790709)
Affinity DataIC50:  3.40nMAssay Description:Binding affinity towards Opioid receptor delta 1 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Northern Colorado

Curated by ChEMBL
LigandPNGBDBM50369571(CHEMBL1790710)
Affinity DataIC50:  4nMAssay Description:Binding affinity towards Opioid receptor mu 1 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Northern Colorado

Curated by ChEMBL
LigandPNGBDBM50369572(CHEMBL1790709)
Affinity DataIC50:  8.20nMAssay Description:Binding affinity towards Opioid receptor mu 1 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069558(2-Amino-N-((S)-1-{[(2-{N'-[2-(2-{(S)-2-[2-amino-3-...)
Affinity DataIC50:  8.80nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069560(Biphalin Analogue | CHEMBL2371080)
Affinity DataIC50:  8.90nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069560(Biphalin Analogue | CHEMBL2371080)
Affinity DataIC50:  8.90nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069563(Biphalin Analogue | CHEMBL2371079)
Affinity DataIC50:  9.30nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069559(Biphalin Analogue | CHEMBL2371057)
Affinity DataIC50:  17nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50:  18nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069562(2-Amino-N-((S)-1-{[((R)-1-{N'-[(R)-2-(2-{(S)-2-[2-...)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069562(2-Amino-N-((S)-1-{[((R)-1-{N'-[(R)-2-(2-{(S)-2-[2-...)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069558(2-Amino-N-((S)-1-{[(2-{N'-[2-(2-{(S)-2-[2-amino-3-...)
Affinity DataIC50:  27nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069561(2-Amino-N-((S)-1-{[((S)-1-{N'-[(S)-2-(2-{(S)-2-[2-...)
Affinity DataIC50:  41nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50:  42nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50:  66nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50:  85nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50069561(2-Amino-N-((S)-1-{[((S)-1-{N'-[(S)-2-(2-{(S)-2-[2-...)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  258nMAssay Description:Opioid receptor activity was evaluated using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  570nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  620nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041666(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...)
Affinity DataIC50:  760nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041666(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...)
Affinity DataIC50:  760nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50:  1.10E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50:  1.20E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50: >2.25E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50:  3.00E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50:  3.30E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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