Affinity DataKi: 0.790nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Compound was tested for binding affinity towards mu opioid receptor in guinea pig brain homogenates using [3H]-CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Compound was tested for binding affinity towards Opioid receptor delta 1 in guinea pig brain homogenates using [3H]-[p-Cl-Phe]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Binding affinity towards Opioid receptor delta 1 was evaluatedMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
University Of Northern Colorado
Curated by ChEMBL
University Of Northern Colorado
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Opioid receptor activity was evaluated using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Binding affinity towards Opioid receptor delta 1 was evaluatedMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity towards Opioid receptor mu 1 was evaluatedMore data for this Ligand-Target Pair
Affinity DataIC50: 8.20nMAssay Description:Binding affinity towards Opioid receptor mu 1 was evaluatedMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibitory concentration required against biological activity of mu opioid receptor from guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration required against biological activity of Opioid receptor delta 1 from mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
University Of Northern Colorado
Curated by ChEMBL
University Of Northern Colorado
Curated by ChEMBL
Affinity DataIC50: 258nMAssay Description:Opioid receptor activity was evaluated using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 760nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 760nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
Affinity DataIC50: >2.25E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair