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Found 12 with Last Name = 'de cupertinis' and Initial = 'a'
TargetEstrogen receptor beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50346462((E)-2-chloro-4,4'-dihydroxybiphenyl-3-carbaldehyde...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]estradiol from human full-length ERbeta receptor by competitive radiometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50346463((E)-2-chloro-3'-fluoro-4,4'-dihydroxybiphenyl-3-ca...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]estradiol from human full-length ERbeta receptor by competitive radiometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50346462((E)-2-chloro-4,4'-dihydroxybiphenyl-3-carbaldehyde...)
Affinity DataEC50:  0.580nMAssay Description:Agonist activity at human full-length ERalpha receptor expressed in human HEC1 cells co-expressing (ERE)2-pS2-luc gene assessed as transcriptional ac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKd:  0.5nMAssay Description:Binding affinity to human full-length ERbeta receptorMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  0.720nMAssay Description:Agonist activity at human full-length ERbeta receptor expressed in human HEC1 cells co-expressing (ERE)2-pS2-luc gene assessed as transcriptional act...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50346464((E)-6-Hydroxy-2,3-bis-(4-hydroxyphenyl)benzaldehyd...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human full-length ERbeta receptor expressed in human HEC1 cells co-expressing (ERE)2-pS2-luc gene assessed as transcriptional act...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50346462((E)-2-chloro-4,4'-dihydroxybiphenyl-3-carbaldehyde...)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at human full-length ERbeta receptor expressed in human HEC1 cells co-expressing (ERE)2-pS2-luc gene assessed as transcriptional act...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50346463((E)-2-chloro-3'-fluoro-4,4'-dihydroxybiphenyl-3-ca...)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human full-length ERbeta receptor expressed in human HEC1 cells co-expressing (ERE)2-pS2-luc gene assessed as transcriptional act...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKd:  0.200nMAssay Description:Binding affinity to human full-length ERalpha receptorMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50346464((E)-6-Hydroxy-2,3-bis-(4-hydroxyphenyl)benzaldehyd...)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human full-length ERalpha receptor expressed in human HEC1 cells co-expressing (ERE)2-pS2-luc gene assessed as transcriptional ac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human full-length ERalpha receptor expressed in human HEC1 cells co-expressing (ERE)2-pS2-luc gene assessed as transcriptional ac...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50346463((E)-2-chloro-3'-fluoro-4,4'-dihydroxybiphenyl-3-ca...)
Affinity DataEC50:  8.40nMAssay Description:Agonist activity at human full-length ERalpha receptor expressed in human HEC1 cells co-expressing (ERE)2-pS2-luc gene assessed as transcriptional ac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed