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Found 1093 with Last Name = 'delisle' and Initial = 'rk'
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104202(US8575145, 79)
Affinity DataIC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104213(US8575145, 120 | US8575145, 121 | US8575145, 150 |...)
Affinity DataIC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104204(US8575145, 81)
Affinity DataIC50:  0.450nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM41535(US8575145, 106 | US8575145, 66)
Affinity DataIC50:  0.5nMAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104229(US8575145, 106)
Affinity DataIC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104162(US8575145, 39)
Affinity DataIC50:  0.550nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104187(US8575145, 64)
Affinity DataIC50:  0.640nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104140(US8575145, 17)
Affinity DataIC50:  0.650nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104186(US8575145, 63)
Affinity DataIC50:  0.650nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104169(US8575145, 46/47/48/49/50 | US8575145, 77 | US8575...)
Affinity DataIC50:  0.700nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104142(US8575145, 19)
Affinity DataIC50:  0.700nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104237(US8575145, 114)
Affinity DataIC50:  0.700nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104221(US8575145, 98)
Affinity DataIC50:  0.700nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104193(US8575145, 70)
Affinity DataIC50:  0.75nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104165(US8575145, 42)
Affinity DataIC50:  0.75nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104188(US8575145, 65)
Affinity DataIC50:  0.800nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104147(US8575145, 24)
Affinity DataIC50:  0.800nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM41535(US8575145, 106 | US8575145, 66)
Affinity DataIC50:  0.800nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104213(US8575145, 120 | US8575145, 121 | US8575145, 150 |...)
Affinity DataIC50:  0.800nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Rattus norvegicus (Rat))
Array Biopharma

US Patent
LigandPNGBDBM104213(US8575145, 120 | US8575145, 121 | US8575145, 150 |...)
Affinity DataIC50:  0.900nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104246(US8575145, 123)
Affinity DataIC50:  0.900nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104169(US8575145, 46/47/48/49/50 | US8575145, 77 | US8575...)
Affinity DataIC50:  0.920nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104190(US8575145, 67)
Affinity DataIC50:  0.950nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104196(US8575145, 73)
Affinity DataIC50:  0.960nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Mus musculus (mouse))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50446319(CHEMBL3109343)
Affinity DataIC50:  1nMAssay Description:Inhibition of PDGF-induced PDGFRbeta phosphorylation in mouse NIH3T3 cells incubated for 1 hr prior to PDGF induction measured after 15 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104215(US8575145, 152 | US8575145, 92 | US8575145, 92/122)
Affinity DataIC50:  1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Mus musculus (mouse))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50446312(CHEMBL3109350)
Affinity DataIC50:  1nMAssay Description:Inhibition of PDGF-induced PDGFRbeta phosphorylation in mouse NIH3T3 cells incubated for 1 hr prior to PDGF induction measured after 15 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104169(US8575145, 46/47/48/49/50 | US8575145, 77 | US8575...)
Affinity DataIC50:  1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104139(US8575145, 16)
Affinity DataIC50:  1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104255(US8575145, 132)
Affinity DataIC50:  1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104248(US8575145, 125)
Affinity DataIC50:  1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104240(US8575145, 117)
Affinity DataIC50:  1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104241(US8575145, 118/119 | US8575145, 149)
Affinity DataIC50:  1.30nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104191(US8575145, 68)
Affinity DataIC50:  1.30nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104226(US8575145, 103)
Affinity DataIC50:  1.40nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104238(US8575145, 115)
Affinity DataIC50:  1.40nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104222(US8575145, 130 | US8575145, 99/100)
Affinity DataIC50:  1.5nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104141(US8575145, 18)
Affinity DataIC50:  1.5nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104256(US8575145, 133)
Affinity DataIC50:  1.60nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104124(US8575145, 1)
Affinity DataIC50:  1.60nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104192(US8575145, 69)
Affinity DataIC50:  1.60nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104233(US8575145, 110)
Affinity DataIC50:  1.90nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Mus musculus (mouse))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50446315(CHEMBL3109347)
Affinity DataIC50:  2nMAssay Description:Inhibition of PDGF-induced PDGFRbeta phosphorylation in mouse NIH3T3 cells incubated for 1 hr prior to PDGF induction measured after 15 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104208(US8575145, 85)
Affinity DataIC50:  2nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Rattus norvegicus (Rat))
Array Biopharma

US Patent
LigandPNGBDBM104141(US8575145, 18)
Affinity DataIC50:  2nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Rattus norvegicus (Rat))
Array Biopharma

US Patent
LigandPNGBDBM104142(US8575145, 19)
Affinity DataIC50:  2nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Rattus norvegicus (Rat))
Array Biopharma

US Patent
LigandPNGBDBM104169(US8575145, 46/47/48/49/50 | US8575145, 77 | US8575...)
Affinity DataIC50:  2nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Rattus norvegicus (Rat))
Array Biopharma

US Patent
LigandPNGBDBM104213(US8575145, 120 | US8575145, 121 | US8575145, 150 |...)
Affinity DataIC50:  2nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Rattus norvegicus (Rat))
Array Biopharma

US Patent
LigandPNGBDBM104222(US8575145, 130 | US8575145, 99/100)
Affinity DataIC50:  2nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50446306(CHEMBL3109340)
Affinity DataIC50:  2nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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