TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario
Curated by ChEMBL
Hospital Regional Universitario
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Positive allosteric modulator activity at GLP-1R in rat INS1 beta-cells assessed potentiation of GLP-1(7-36)NH2 induced insulin secretion at 0.1 nM i...More data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario
Curated by ChEMBL
Hospital Regional Universitario
Curated by ChEMBL
Affinity DataEC50: 0.25nMAssay Description:Positive allosteric modulator activity at GLP-1R in rat INS1 beta-cells assessed potentiation of GLP-1(7-36)NH2 induced insulin secretion incubated f...More data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario
Curated by ChEMBL
Hospital Regional Universitario
Curated by ChEMBL
Affinity DataEC50: 0.00800nMAssay Description:Positive allosteric modulator activity at GLP-1R in rat INS1 beta-cells assessed potentiation of GLP-1(7-36)NH2 induced insulin secretion incubated f...More data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Hospital Regional Universitario
Curated by ChEMBL
Hospital Regional Universitario
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Positive allosteric modulator activity at human GLP-1R expressed in HEK293 cells assessed as activation of calcium fluxMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Hospital Regional Universitario
Curated by ChEMBL
Hospital Regional Universitario
Curated by ChEMBL
Affinity DataEC50: 0.100nMAssay Description:Positive allosteric modulator activity at human GLP-1R expressed in HEK293 cells assessed as potentiation of GLP-1(7-36)NH2 induced cAMP accumulation...More data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Hospital Regional Universitario
Curated by ChEMBL
Hospital Regional Universitario
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Positive allosteric modulator activity at human GLP-1R expressed in HEK293 cells assessed as activation of calcium fluxMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Positive allosteric modulation of human 5-HT2C receptor expressed in human HeLa-K1 cells assessed as potentiation of 5-HT-induced inositol monophosph...More data for this Ligand-Target Pair