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Found 24 with Last Name = 'dijkgraaf' and Initial = 'i'
TargetSomatostatin receptor type 2(RAT)
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50318385(2-(4-{[(2-{[(3-{[1-(5-{[(1R)-1-{[(4R,7S,10S,13R,16...)
Affinity DataIC50:  1.32nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363984(CHEMBL1949730)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363974(CHEMBL1949739)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50318386(2-[7-({[2-({[3,5-bis({[1-(5-{[(1R)-1-{[(4R,7S,10S,...)
Affinity DataIC50:  2.45nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50318388((4R,7S,10S,13R,16S,19R)-10-(4-aminobutyl)-N-[(2R,3...)
Affinity DataIC50:  2.45nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363973(CHEMBL1949738)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363969(CHEMBL1949734)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363975(CHEMBL1949740)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363972(CHEMBL1949737)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363978(CHEMBL1949885)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363986(CHEMBL1949731)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363977(CHEMBL1949884)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363971(CHEMBL1949736)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363979(CHEMBL1949886)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50318387(CHEMBL1099306)
Affinity DataIC50:  14nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363983(CHEMBL1949890)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363970(CHEMBL1949735)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363981(CHEMBL1949888)
Affinity DataIC50:  31nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363976(CHEMBL1949741)
Affinity DataIC50:  33nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363982(CHEMBL1949889)
Affinity DataIC50:  39nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363987(CHEMBL1949732)
Affinity DataIC50:  60nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363968(CHEMBL1949733)
Affinity DataIC50:  67nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363980(CHEMBL1949887)
Affinity DataIC50:  98nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363985(CHEMBL1949675)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed