Affinity DataIC50: 2.90nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
Target InfoGoogleScholar
Affinity DataIC50: 4.20nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
Target InfoGoogleScholar
Affinity DataIC50: 14nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Compound was evaluated for its inhibitory activity against Leucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
Target InfoGoogleScholar
Affinity DataIC50: 25nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
Target InfoGoogleScholar
Affinity DataIC50: 30nMAssay Description:Compound was evaluated for its inhibitory activity against VRS (valyl tRNA synthetase) from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
Target InfoGoogleScholar
Affinity DataIC50: 120nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Compound was evaluated for its inhibitory activity against VRS (valyl tRNA synthetase) from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Compound was evaluated for its inhibitory activity against VRS (valyl tRNA synthetase) from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
Target InfoGoogleScholar
Affinity DataIC50: 910nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.55E+3nMAssay Description:Compound was evaluated for its inhibitory activity against Leucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Compound was evaluated for its inhibitory activity against Leucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.27E+3nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
Target InfoGoogleScholar
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.46E+4nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
Affinity DataIC50: 2.23E+4nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
Target InfoGoogleScholar
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 7.10E+4nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 7.60E+4nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.20E+5nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.60E+5nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.80E+5nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.86E+5nMAssay Description:Compound was evaluated for its inhibitory activity against Leucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 2.00E+5nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 2.10E+5nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 2.90E+5nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 3.50E+5nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 3.70E+5nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 3.70E+5nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 5.00E+5nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 5.60E+5nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 6.00E+5nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 9.80E+5nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.10E+6nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.10E+6nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.10E+6nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.10E+6nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair