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Found 32 with Last Name = 'el mourabit' and Initial = 'h'
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50135601((S,E)-N1-(3-(1H-indol-3-yl)-1-(methylamino)-1-oxop...)
Affinity DataIC50:  9.20nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50135601((S,E)-N1-(3-(1H-indol-3-yl)-1-(methylamino)-1-oxop...)
Affinity DataIC50:  10nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  13nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50135601((S,E)-N1-(3-(1H-indol-3-yl)-1-(methylamino)-1-oxop...)
Affinity DataIC50:  17nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50135601((S,E)-N1-(3-(1H-indol-3-yl)-1-(methylamino)-1-oxop...)
Affinity DataIC50:  18nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213416((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-3-phenylprop-2...)
Affinity DataIC50:  38nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213419((2E)-3-(N-hydroxycarbamoyl)-2-(3-phenylpropylidene...)
Affinity DataIC50:  45nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213418((2E)-3-(N-hydroxycarbamoyl)-2-heptylidenepropionyl...)
Affinity DataIC50:  101nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213416((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-3-phenylprop-2...)
Affinity DataIC50:  120nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213418((2E)-3-(N-hydroxycarbamoyl)-2-heptylidenepropionyl...)
Affinity DataIC50:  122nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213418((2E)-3-(N-hydroxycarbamoyl)-2-heptylidenepropionyl...)
Affinity DataIC50:  123nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50135601((S,E)-N1-(3-(1H-indol-3-yl)-1-(methylamino)-1-oxop...)
Affinity DataIC50:  179nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213419((2E)-3-(N-hydroxycarbamoyl)-2-(3-phenylpropylidene...)
Affinity DataIC50:  280nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213417((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-but-2-en-1-yli...)
Affinity DataIC50:  913nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213417((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-but-2-en-1-yli...)
Affinity DataIC50:  974nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213417((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-but-2-en-1-yli...)
Affinity DataIC50:  984nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213416((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-3-phenylprop-2...)
Affinity DataIC50:  1.24E+3nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213419((2E)-3-(N-hydroxycarbamoyl)-2-(3-phenylpropylidene...)
Affinity DataIC50:  1.92E+3nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213416((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-3-phenylprop-2...)
Affinity DataIC50:  2.49E+3nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213418((2E)-3-(N-hydroxycarbamoyl)-2-heptylidenepropionyl...)
Affinity DataIC50:  2.66E+3nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213417((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-but-2-en-1-yli...)
Affinity DataIC50:  8.61E+3nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213419((2E)-3-(N-hydroxycarbamoyl)-2-(3-phenylpropylidene...)
Affinity DataIC50:  9.13E+3nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213416((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-3-phenylprop-2...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213418((2E)-3-(N-hydroxycarbamoyl)-2-heptylidenepropionyl...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213419((2E)-3-(N-hydroxycarbamoyl)-2-(3-phenylpropylidene...)
Affinity DataIC50:  5.31E+4nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213417((2E)-3-(N-hydroxycarbamoyl)-2-[(2E)-but-2-en-1-yli...)
Affinity DataIC50:  7.85E+4nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213418((2E)-3-(N-hydroxycarbamoyl)-2-heptylidenepropionyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213418((2E)-3-(N-hydroxycarbamoyl)-2-heptylidenepropionyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed